Ballicules.com

Drug classes and tags

5-Alpha-reductase inhibitors (2)

FinasterideDutasteride

5-HT2A receptor agonists (9)

Lysergic acid diethylamidePsilocinN,N-dimethyl­ tryptamineMescalineErgotaminemCPPMethylenedioxy­ methamphetamineSerotoninPsilocybin

ADHD non-stimulants (8)

AtomoxetineViloxazineGuanfacineClonidineCentanafadineClonidine ERClonidine ER suspensionGuanfacine ER

Abortifacients (3)

MifepristoneMisoprostolMethotrexate

Acid-suppressing drugs (20)

OmeprazolePantoprazoleFamotidineEsomeprazoleSucralfateLansoprazoleDexlansoprazoleRabeprazoleCimetidineMisoprostolNizatidineCalcium carbonateMg hydroxideAprepitantNetupitantAl/Mg antacidAluminum hydroxideBismuth subsalicylateRanitidineVonoprazan

Acne medications (9)

TretinoinDapsoneIsotretinoinClindamycinDoxycyclineMinocyclineNorgestimateSpironolactoneTazarotene

Acute interstitial nephritis (22)

IbuprofenNaproxenDiclofenacIndomethacinKetorolacMesalamineMeloxicamCelecoxibNabumetoneEtodolacSulindacPiroxicamFlurbiprofenOxaprozinDiflunisalSalsalateKetoprofenMefenamic acidDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchMesalamine DR

Adenosine receptor agonists (2)

AdenosineRegadenoson

Adrenergic agonists (31)

EpinephrineNorepinephrinePhenylephrineDopamineDobutamineAlbuterolClonidineGuanfacineMidodrinePseudoephedrineTizanidineBrimonidineDihydro­ ergotamineOxymetazolineLofexidineErgotamineDexmedetomidineGuanabenzMethyldopaXylazineDroxidopaFormoterolIsoproterenolSalmeterolTerbutalineAlbuterol nebulizerClonidine ERClonidine ER suspensionDesglymidodrineDexmedetomidine sublingualGuanfacine ER

Adrenocorticotropic hormone (ACTH) analogs (1)

Corticotropin

Alcohol use disorder medications (5)

NaltrexoneAcamprosateDisulfiramNalmefeneNaltrexone ER injection

Alkylating agents (5)

CyclophosphamideIfosfamideProcarbazinePhosphoramide mustardTemozolomide

Alpha-1 blockers (80)

PrazosinDoxazosinTerazosinTamsulosinAlfuzosinSilodosinPhenoxybenzaminePhentolamineCarvedilolLabetalolTrazodoneQuetiapineMirtazapineCyclobenzaprineHydroxyzine HClAripiprazoleRisperidoneOlanzapineAmitriptylinePromethazineDoxepinClozapineHaloperidolPaliperidoneBrexpiprazoleChlorpromazineFluphenazineCyproheptadinePerphenazineImipramineClomipramineLumateperoneAsenapineIloperidoneTrifluoperazineThioridazineThiothixeneMilsaperidoneProtriptylineNefazodoneAmoxapineTrimipramineDoxylamine8-OH-AmoxapineDehydro­ aripiprazole(Desmethyl-) mirtazapineDesmethyl­ clomipramineHydroxy­ nefazodoneMianserinNorclozapineNordoxepinNorquetiapineDesipramineDroperidolLoxapineLurasidoneMaprotilineMolindonePimozideProchlorperazineZiprasidoneAripiprazole lauroxil LAIAripiprazole lauroxil LAIAripiprazole monohydrate LAIAripiprazole monohydrate LAIAsenapine transdermalClozapine ODTClozapine oral suspensionDoxepin low-dose (insomnia)Fluphenazine decanoate LAIHaloperidol decanoate LAIHaloperidol injectionHydroxyzine IMLoxapine inhaledPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIQuetiapine XRZiprasidone IM

Alpha-2 agonists (16)

ClonidineGuanfacineDexmedetomidineMethyldopaTizanidineBrimonidineOxymetazolineLofexidineGuanabenzNorepinephrineXylazineMirtazapineClonidine ERClonidine ER suspensionDexmedetomidine sublingualGuanfacine ER

Alpha-2 antagonists (5)

1-PPMianserinPhenoxybenzaminePhentolamineYohimbine

Alpha-glucosidase inhibitors (2)

AcarboseVoglibose

Aminoglycosides (4)

GentamicinTobramycinNeomycinAmikacin

Ammonia-lowering agents (4)

RifaximinNeomycinLactuloseLevocarnitine

Amphetamines (14)

AmphetamineDextro­ amphetamineMethamphetamineLisdexamfetaminePhentermineAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)Dextroamphetamine IR tabletsDextroamphetamine oral solutionDextroamphetamine patchDextroamphetamine spansuleMixed amphetamine salts (triple-bead)Mixed amphetamine salts XR

Amylin analogs (1)

Pramlintide

Anabolic steroids (3)

TestosteroneDanazolTestosterone cypionate

Analgesics (129)

TramadolMeloxicamOxycodoneDiclofenacIbuprofenCelecoxibNaproxenMorphineKetorolacNaloxoneFentanylHydromorphoneLoperamideDiphenoxylateNabumetoneMethadoneBuprenorphineSuzetrigineNaltrexoneSuvorexantBromfenacNaloxegolEtodolacIndomethacinSulindacTapentadolMisoprostolMethylnaltrexonePiroxicamHydrocodoneLemborexantPhenazopyridineOxymorphoneEluxadolineDaridorexantButorphanolNaldemedineFlurbiprofenOxaprozinCodeineDiflunisalPentazocineSalsalateLevorphanolApomorphineKetoprofenMeperidineNalbuphineLofexidineDifenoxinAcetaminophenMefenamic acidZiconotideNalmefeneAlfentanilAlvimopanAspirinBeta-endorphinDifelikefalinDynorphinEndomorphinsEnkephalinHeroinMitragynineNociceptinO-desmethyl- tramadolOliceridineOrexin AR-MethadoneRemifentanilS-MethadoneSalicylateSalvinorin ASamidorphanSeltorexantSufentanilTianeptineAlmotriptanArticaineAtogepantBupivacaineCapsaicinDihydro­ ergotamineEletriptanErgotamineFenoprofenFrovatriptanLasmiditanLidocaineIV lipid emulsionMeclofenamateMepivacaineMetaxaloneMethocarbamolNaratriptanOrphenadrinePrilocaineProcaineRimegepantRizatriptanRopivacaineSumatriptanTetracaineTolmetinUbrogepantZavegepantZolmitriptan6-MNABuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERLidocaine injectionMorphine ER capsulesMorphine ER tabletsNaloxone nasal sprayNaltrexone ER injectionOxycodone CRSulindac sulfideSumatriptan SC injectionSumatriptan nasalTramadol ER

Anaphylaxis-associated medications (16)

Penicillin VAmoxicillinAmpicillinCefazolinCeftriaxoneVancomycinInfliximabPaclitaxelCisplatinSuccinylcholineRocuroniumAtracuriumAmphotericin BIcatibantOmalizumabProtamine sulfate

Androgens (4)

TestosteroneDanazolDehydroepi­ androsteroneTestosterone cypionate

Anesthetics (23)

PropofolEtomidateKetamineThiopentalMethohexitalSevofluraneIsofluraneDesfluraneNitrous oxideLidocaineBupivacaineRopivacaineMepivacainePrilocaineProcaineTetracaineArticaineCocaineMidazolamRemifentanilSufentanilAlfentanilLidocaine injection

Angiotensin receptor blockers (ARBs) (8)

LosartanValsartanIrbesartanCandesartanOlmesartanTelmisartanEprosartanAzilsartan

Angiotensin receptor–neprilysin inhibitors (ARNIs) (2)

SacubitrilValsartan

Angiotensin-converting enzyme (ACE) inhibitors (11)

LisinoprilBenazeprilEnalaprilRamiprilFosinoprilCaptoprilQuinaprilTrandolaprilMoexiprilPerindoprilEnalaprilat

Anthelmintics (2)

AlbendazoleIvermectin

Anti-inflammatory drugs (58)

PrednisoneFluticasoneMeloxicamDiclofenacIbuprofenTriamcinoloneMethyl­ prednisoloneCelecoxibPrednisoloneNaproxenHydrocortisoneClobetasolMethotrexateTiotropiumIpratropiumKetorolacDexamethasoneColchicineMometasoneUmeclidiniumBetamethasoneFluocinonideNabumetoneSulfasalazineBudesonideLeflunomideFludrocortisoneFluorometholoneLoteprednolBromfenacEtodolacIndomethacinHalobetasolSulindacBeclomethasoneMisoprostolFlunisolidePiroxicamFlurbiprofenOxaprozinAclidiniumDiflunisalSalsalateKetoprofenPenicillamineMefenamic acidAspirinSalicylateFenoprofenMeclofenamateTolmetinDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchFluticasone nasalHydrocortisone topicalIpratropium nasalTriamcinolone injection

Anti-obesity drugs (17)

SemaglutideDulaglutideTirzepatideLiraglutideExenatidePhentermineLorcaserinOrforglipronPhendimetrazineRetatrutideRimonabantSetmelanotideLiraglutide (obesity)Semaglutide (obesity)Semaglutide oralSemaglutide oral (obesity)Tirzepatide (obesity)

Antiandrogens (7)

BicalutamideEnzalutamideApalutamideAbirateroneFinasterideDutasterideSpironolactone

Antianemic drugs (11)

Ferric citrateFolic acidCyanocobalaminHydroxocobalaminAdenosylcobalaminFilgrastimDarbepoetin alfaEpoetin alfaFerrous sulfateRoxadustatVadadustat

Antianginal drugs (19)

AmlodipineMetoprololAtenololDiltiazemIsosorbide mononitrateNifedipineNitroglycerinVerapamilRanolazineIsosorbide dinitrateNadololVericiguatNicardipineAmyl nitriteIvabradineDiltiazem ERMetoprolol succinate ERNifedipine ER (GITS)Verapamil ER

Antiarrhythmic drugs (Class I) (17)

LidocaineFlecainideQuinidinePropafenoneMexiletineHydroquinidineEncainideProcainamideTocainideDisopyramideAprindinePilsicainideAjmalineEthacizineCibenzolineMoricizineLidocaine injection

Antiarrhythmic drugs (Class IA) (6)

QuinidineHydroquinidineProcainamideDisopyramideAjmalineCibenzoline

Antiarrhythmic drugs (Class IB) (5)

LidocaineMexiletineTocainideAprindineLidocaine injection

Antiarrhythmic drugs (Class IC) (6)

FlecainidePropafenoneEncainidePilsicainideEthacizineMoricizine

Antiarrhythmic drugs (Class II) (11)

PropranololMetoprololEsmololAtenololAcebutololNadololBisoprololLabetalolSotalolMetoprolol succinate ERPropranolol ER

Antiarrhythmic drugs (Class III) (5)

AmiodaroneDronedaroneSotalolDofetilideIbutilide

Antiarrhythmic drugs (Class IV) (5)

VerapamilDiltiazemDiltiazem EREtripamilVerapamil ER

Antiarrhythmic drugs (all) (41)

PropranololAmiodaroneVerapamilLidocaineFlecainideQuinidineMetoprololDiltiazemDronedaronePropafenoneMexiletineHydroquinidineSotalolEncainideEsmololProcainamideTocainideAtenololDofetilideDisopyramideAprindinePilsicainideAcebutololAjmalineEthacizineIbutilideNadololCibenzolineMoricizineBisoprololLabetalolAdenosineDigoxinMagnesiumAtropineAtropine eyedropsDiltiazem ERLidocaine injectionMetoprolol succinate ERPropranolol ERVerapamil ER

Antibacterial drugs (89)

AmoxicillinAzithromycinCephalexinCiprofloxacinMupirocinLevofloxacinClindamycinMetronidazoleCefdinirDoxycyclineErythromycinOfloxacinMoxifloxacinMethenamine hippurateSilver sulfadiazineSulfasalazineCefadroxilCefpodoximeGentamicinRifaximinVancomycinMinocyclineCeftriaxoneTobramycinClarithromycinTrimethoprimErtapenemDaptomycinLinezolidBalsalazideRifampinFosfomycinCefepimeDapsoneMeropenemCefazolinEthambutolNeomycinTetracyclineIsoniazidFidaxomicinDicloxacillinAmpicillinCeftazidimeCefiximeRifabutinAmikacinDemeclocyclineMethenamine mandelatePenicillin VAztreonamNafcillinOxacillinNitrofurantoinRifapentinePyrimethaminePolymyxin BCefuroximeCycloserineChloramphenicolCloxacillinEnoxacinImipenemMethicillinSulfamethoxazoleTelithromycinCefotaximeCefoxitinCeftarolinePenicillin GPiperacillinTedizolidBedaquilineCefaclorCefprozilCeftizoximeCephradineCilastatinDelafloxacinFlucloxacillinGatifloxacinGemifloxacinGepotidacinNemonoxacinNorfloxacinPyrazinamideSparfloxacinTicarcillinZoliflodacin

Antibodies (25)

EvolocumabAdalimumabAlirocumabDupilumabDenosumabTocilizumabSarilumabInfliximabErenumabFremanezumabGalcanezumabIdarucizumabRomosozumabSiltuximabEtanerceptNatalizumabNivolumabPembrolizumabRituximabAnifrolumabBelimumabDonanemabEfgartigimodLecanemabNirsevimab

Anticoagulants (21)

ApixabanClopidogrelRivaroxabanWarfarinTicagrelorDabigatranEnoxaparinPrasugrelTafamidisHeparinPentosan polysulfateTranexamic acidFondaparinuxEdoxabanAndexanet alfaIdarucizumabProtamine sulfateTiclopidineArgatrobanBetrixabanBivalirudin

Antidepressants (50)

SertralineEscitalopramFluoxetineCitalopramParoxetineFluvoxamineVenlafaxineDuloxetineDesvenlafaxineBupropionMirtazapineVortioxetineVilazodoneTrazodoneNefazodoneAmitriptylineImipramineClomipramineNortriptylineDesipramineDoxepinPhenelzineTranylcypromineIsocarboxazidEsketamineZuranoloneMilnacipranLevomilnacipranDextromethorphanGepironeProtriptylineAmoxapineTrimipramineKetamineMianserinSt John's wortTianeptineReboxetineViloxazineBupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERDoxepin low-dose (insomnia)Fluvoxamine CRMaprotilineMoclobemideParoxetine CRVenlafaxine XR

Antidiarrheals (7)

LoperamideDiphenoxylateEluxadolineDifenoxinAlosetronCholestyramineRifaximin

Antidotes and chelators (36)

NaloxoneCyproheptadineDantroleneDeferasiroxFlumazenilDeferiproneDeferoxaminePhysostigmineN-acetylcysteine (NAC)PhytonadioneAndexanet alfaDigoxin immune FabDimercaprolEdetate calcium disodiumGlucarpidaseIdarucizumabIV lipid emulsionMethylene bluePenicillaminePralidoximeProtamine sulfatePrussian blueTrientineAcetylcysteineActivated charcoalAmyl nitriteAtropineAtropine eyedropsDexrazoxaneFomepizoleGlucagonHydroxocobalaminMesnaNalmefeneNaloxone nasal spraySodium thiosulfate

Antiemetics (18)

OndansetronMeclizinePromethazineMetoclopramideProchlorperazineScopolamineDronabinolAprepitantGranisetronRolapitantDoxylamineTrimethobenzamideAmisulprideNabiloneDimenhydrinateDomperidoneNetupitantPalonosetron

Antiepileptic drugs (AEDs) (49)

GabapentinMagnesiumClonazepamPregabalinLevetiracetamLamotrigineTopiramateCarbamazepinePrimidoneOxcarbazepineLacosamidePhenobarbitalZonisamideClobazamPhenytoinBrivaracetamEslicarbazepineCenobamatePerampanelCannabidiolGabapentin enacarbilRufinamideFelbamateTiagabineEthosuximideMethsuximideVigabatrinFenfluramineStiripentolFosphenytoinGanaxolonePentobarbitalEzogabinePyridoxal-5'- phosphateValproic acidKynurenic acidLevocarnitineCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRDivalproex DRDivalproex ERDivalproex sprinkleLacosamide ERLamotrigine XROxcarbazepine XRTopiramate ERTopiramate ER (sprinkle)Valproate sodium IV

Antifibrinolytics (1)

Tranexamic acid

Antifungal drugs (17)

NystatinKetoconazoleFluconazoleClotrimazoleCiclopiroxTerbinafineVoriconazoleItraconazolePosaconazoleIsavuconazoniumMicafunginGriseofulvinMiconazoleAmphotericin BIsavuconazoleFlucytosineCaspofungin

Antiglaucoma drugs (19)

LatanoprostClonidineTimololBrimonidineBimatoprostDorzolamideTravoprostNetarsudilAcetazolamidePilocarpineBrinzolamideMethazolamideBetaxololCarteololMannitolAceclidineCarbacholClonidine ERClonidine ER suspension

Antigout drugs (6)

LosartanAllopurinolColchicineFebuxostatProbenecidLesinurad

Antihistamines (28)

DiphenhydramineDimenhydrinateDoxylamineChlorpheniramineBrompheniramineHydroxyzine HClMeclizinePromethazineCyproheptadineKetotifenCetirizineLevocetirizineLoratadineDesloratadineFexofenadineAzelastineOlopatadineFamotidineCimetidineNizatidineCyclobenzaprinePitolisantThiothixeneTrifluoperazineDiphenhydramine injectionHydroxyzine IMHydroxyzine pamoatePromethazine injection

Antihypertensive drugs (75)

AmlodipineLisinoprilLosartanMetoprololHydrochloro­ thiazideCarvedilolAtenololDiltiazemHydralazineValsartanPropranololNifedipineOlmesartanChlorthalidoneTorsemideIrbesartanBenazeprilDoxazosinEnalaprilVerapamilRamiprilNebivololPrazosinSotalolTelmisartanLabetalolBisoprololCandesartanIndapamideFelodipineNadololGuanfacineFosinoprilAzilsartanMacitentanCaptoprilAcebutololAmbrisentanQuinaprilTrandolaprilBaxdrostatRiociguatSelexipagAliskirenPindololMoexiprilCarteololPerindoprilTreprostinilEthacrynic acidNisoldipineBosentanIsradipineNicardipineNimodipineEpoprostenolChlorothiazideEprosartanGuanabenzMethyldopaReserpineEXP3174 (E-3174)EXP3179NitroprussideSacubitrilAprocitentanDiltiazem EREnalaprilatGuanfacine ERMetoprolol succinate ERMoxonidineNifedipine ER (GITS)Propranolol ERRilmenidineVerapamil ER

Antimalarial drugs (5)

Hydroxy­ chloroquineAtovaquoneMefloquineChloroquinePyrimethamine

Antimetabolites (13)

MethotrexateFluorouracilCapecitabineMercaptopurineAzathioprineMycophenolate mofetilHydroxyureaLeflunomideTeriflunomidePyrimethamineTrimethoprimFlucytosineRibavirin

Antimicrobial drugs—topical (14)

NystatinMupirocinClotrimazoleCiclopiroxTerbinafineSilver sulfadiazineRifaximinMiconazoleMetronidazoleNeomycinPermethrinPolymyxin BBenzoyl peroxideChlorhexidine

Antimicrobials (178)

AmoxicillinAzithromycinCephalexinCiprofloxacinNystatinKetoconazoleFluconazoleMupirocinValacyclovirLevofloxacinClindamycinMetronidazoleCefdinirAcyclovirDoxycyclineErythromycinOfloxacinMoxifloxacinClotrimazoleCiclopiroxTerbinafineSilver sulfadiazineAmantadineCefadroxilCefpodoximeOseltamivirGentamicinRifaximinMolnupiravirVancomycinMinocyclineCeftriaxoneDolutegravirTobramycinClarithromycinTrimethoprimErtapenemDaptomycinFamciclovirEntecavirLinezolidRifampinValganciclovirCefepimeDapsoneMeropenemTenofovirCefazolinDarunavirRaltegravirEthambutolIvermectinNeomycinRitonavirProbenecidTetracyclineLamivudineDoravirineVoriconazoleIsoniazidItraconazolePosaconazoleEtravirineDicloxacillinAmpicillinAbacavirGanciclovirMaravirocRilpivirineCeftazidimeIsavuconazoniumCefiximeAtazanavirRifabutinEfavirenzNevirapineMicafunginAmikacinDemeclocyclineFostemsavirLetermovirEmtricitabineBaloxavir marboxilGriseofulvinPenicillin VAztreonamNafcillinOxacillinNitrofurantoinCabotegravirMiconazoleRifapentineCobicistatNelfinavirPyrimethamineRemdesivirPolymyxin BCefuroximeCidofovirPentamidineAmphotericin BCycloserineBictegravirChloramphenicolDasabuvirElvitegravirEnoxacinGlecaprevirIndinavirIsavuconazoleLedipasvirLopinavirNirmatrelvirOmbitasvirParitaprevirPibrentasvirSaquinavirSulfamethoxazoleVelpatasvirAlbendazoleAtovaquoneBalsalazideCefotaximeCefoxitinCeftarolineClavulanateCloxacillinFidaxomicinFlucytosineFosfomycinHydroxy­ chloroquineImipenemMefloquineMethenamine hippurateMethenamine mandelateMethicillinPenicillin GPermethrinPiperacillinSulfasalazineTedizolidTelithromycinAmantadine ERAvibactamBedaquilineBemnifosbuvirCaspofunginCefaclorCefprozilCeftizoximeCephradineCilastatinDaclatasvirDelafloxacinDidanosineElbasvirFlucloxacillinGatifloxacinGemifloxacinGepotidacinGrazoprevirIslatravirLenacapavir (PrEP)MaribavirNemonoxacinNorfloxacinPyrazinamideRelebactamSimeprevirSofosbuvirSparfloxacinSulbactamTazobactamTenofovir alafenamideTicarcillinVaborbactamZidovudineZoliflodacin

Antimigraine drugs—acute (17)

SumatriptanRizatriptanRimegepantUbrogepantAtogepantNaratriptanEletriptanZolmitriptanDihydro­ ergotamineLasmiditanFrovatriptanAlmotriptanZavegepantErgotamineButalbitalSumatriptan SC injectionSumatriptan nasal

Antimigraine drugs—preventive (19)

PropranololTopiramateCandesartanRimegepantAtogepantErenumabFremanezumabGalcanezumabValproic acidAmitriptylineRiboflavinBotulinum toxinDivalproex DRDivalproex ERDivalproex sprinklePropranolol ERTopiramate ERTopiramate ER (sprinkle)Valproate sodium IV

Antimuscarinic drugs (72)

OxybutyninDicyclomineTiotropiumIpratropiumBenztropineSolifenacinUmeclidiniumTolterodineTrospiumScopolamineGlycopyrrolateTrihexyphenidylFesoterodineAtropineDarifenacinHyoscyamineCyclopentolateAclidiniumTropicamideAmitriptylineImipramineDisopyramideTrimipramineNortriptylineOlanzapinePromethazineDoxepinClozapineChlorpromazineClomipramineOrphenadrineDiphenhydramineThioridazineDoxylamineQuetiapineCyclobenzaprineCyproheptadineCarbamazepineProtriptylineBrompheniramineChlorpheniramineDesmethyl­ clomipramineDimenhydrinateNordoxepinNorquetiapineDesipramineLoxapineMaprotilineParoxetinePerphenazineProchlorperazineRevefenacinAmoxapine5-HMTAtropine eyedropsCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRChlorpromazine injectionClozapine ODTClozapine oral suspensionDiphenhydramine injectionDoxepin low-dose (insomnia)Glycopyrrolate inhaledIpratropium nasalLoxapine inhaledOlanzapine IMOlanzapine pamoate LAIOxybutynin ERParoxetine CRPromethazine injectionQuetiapine XR

Antimycobacterial drugs (10)

RifampinEthambutolIsoniazidRifabutinRifapentineCycloserineAmikacinDapsoneBedaquilinePyrazinamide

Antineoplastic drugs (67)

MethotrexateFluorouracilHydroxyureaIbrutinibRuxolitinibPalbociclibImatinibLeucovorinVenetoclaxAcalabrutinibOsimertinibZanubrutinibAbemaciclibMercaptopurineEverolimusDasatinibSirolimusOlaparibRibociclibNilotinibBosutinibTrametinibDabrafenibAlectinibAprepitantNiraparibSotorasibGranisetronRegorafenibErlotinibBexaroteneCyclophosphamideTucatinibLorlatinibFilgrastimCrizotinibPaclitaxelVemurafenibMitotaneIdelalisibCisplatinRolapitantVincristineCeritinibCapecitabineVorinostatVandetanibTopotecanTemsirolimusRomidepsinNabiloneIfosfamideNetupitantBelinostatBleomycinBortezomibCollagenase clostridium histolyticumDoxorubicinEtoposideGivinostatIrinotecanNivolumabPanobinostatPembrolizumabRituximabPhosphoramide mustardTirbanibulin

Antiparasitic drugs (10)

Hydroxy­ chloroquineMetronidazoleAtovaquoneIvermectinMefloquineAlbendazoleChloroquinePyrimethaminePentamidinePermethrin

Antiplatelet drugs (20)

ClopidogrelTicagrelorCilostazolPrasugrelDipyridamoleAspirinTiclopidineAndexanet alfaApixabanDabigatranEnoxaparinFondaparinuxHeparinIdarucizumabProtamine sulfateRivaroxabanTafamidisTranexamic acidWarfarinClopidogrel active metabolite

Antiprotozoal drugs (7)

Hydroxy­ chloroquineMetronidazoleAtovaquoneMefloquineChloroquinePyrimethaminePentamidine

Antipruritic drugs (10)

Hydroxyzine HClPromethazineDiphenhydramineObeticholic acidDifelikefalinCetirizineCholestyramineDoxepinDoxepin low-dose (insomnia)Hydroxyzine IM

Antipsychotics (58)

ClozapineRisperidoneOlanzapineQuetiapineZiprasidoneAripiprazolePaliperidoneAsenapineIloperidoneLurasidoneBrexpiprazoleCariprazineLumateperonePimavanserinAmisulprideSulpirideMilsaperidoneHaloperidolChlorpromazineFluphenazinePerphenazineTrifluoperazineThioridazineThiothixeneLoxapineMolindonePimozideProchlorperazineDroperidolFlupentixol7-OH loxapine8-OH-AmoxapineAmoxapineDehydro­ aripiprazoleDesmethyl­ cariprazineDidesmethyl­ cariprazineNorclozapineXanomelineAripiprazole lauroxil LAIAripiprazole lauroxil LAIAripiprazole monohydrate LAIAripiprazole monohydrate LAIAsenapine transdermalChlorpromazine injectionClozapine ODTClozapine oral suspensionFluphenazine decanoate LAIHaloperidol decanoate LAIHaloperidol injectionLoxapine inhaledMelperoneOlanzapine IMPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIQuetiapine XRZiprasidone IM

Antirheumatic drugs (15)

Hydroxy­ chloroquineMethotrexateAdalimumabSulfasalazineLeflunomideEtanerceptTofacitinibUpadacitinibTocilizumabSarilumabInfliximabDiflunisalSalsalatePenicillamineRituximab

Antiseptics and disinfectants (5)

Methenamine hippurateMethenamine mandelateSilver sulfadiazineBenzoyl peroxideChlorhexidine

Antispasmodics (7)

DicyclomineMetoclopramideGlycopyrrolateHyoscyamineAlosetronScopolamineGlycopyrrolate inhaled

Antithyroid drugs (2)

MethimazolePropylthiouracil

Antitumor antibiotics (2)

BleomycinDoxorubicin

Antitussives (5)

BenzonatateDextromethorphanCodeineGuaifenesinHydrocodone

Antiviral drugs (68)

ValacyclovirAcyclovirSilver sulfadiazineAmantadineOseltamivirMolnupiravirDolutegravirFamciclovirEntecavirValganciclovirTenofovirDarunavirRaltegravirRitonavirLamivudineDoravirineEtravirineAbacavirGanciclovirMaravirocRilpivirineAtazanavirEfavirenzNevirapineFostemsavirLetermovirEmtricitabineBaloxavir marboxilCabotegravirCobicistatNelfinavirRemdesivirCidofovirPentamidineBictegravirDasabuvirElvitegravirGlecaprevirIndinavirLedipasvirLopinavirNirmatrelvirOmbitasvirParitaprevirPibrentasvirSaquinavirVelpatasvirAdefovirFoscarnetLenacapavirNitric oxidePeginterferon alfaRibavirinAmantadine ERBemnifosbuvirDaclatasvirDidanosineElbasvirGrazoprevirIslatravirLenacapavir (PrEP)MaribavirNirsevimabPenciclovirSimeprevirSofosbuvirTenofovir alafenamideZidovudine

Anxiolytics (28)

BuspironeAlprazolamLorazepamDiazepamClonazepamChlordiazepoxideOxazepamClorazepateHydroxyzine HClSertralineEscitalopramParoxetineFluoxetineFluvoxamineVenlafaxineDuloxetinePregabalinGabapentinPropranololLavenderGepironeAlprazolam XRFluvoxamine CRHydroxyzine IMLorazepam injectionParoxetine CRPropranolol ERVenlafaxine XR

Aromatase inhibitors (3)

AnastrozoleLetrozoleExemestane

Asthma biologics (6)

DupilumabOmalizumabTralokinumabBenralizumabMepolizumabTezepelumab

Attention-deficit/hyperactivity disorder (ADHD) medications (40)

MethylphenidateDex­ methylphenidateAmphetamineDextro­ amphetamineLisdexamfetamineMethamphetamineAtomoxetineViloxazineGuanfacineClonidineCentanafadineModafinilAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)Clonidine ERClonidine ER suspensionDexmethylphenidate XRDextroamphetamine IR tabletsDextroamphetamine oral solutionDextroamphetamine patchDextroamphetamine spansuleGuanfacine ERMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchMixed amphetamine salts (triple-bead)Mixed amphetamine salts XRSerdexmethylphenidate

Azole antifungals (9)

KetoconazoleFluconazoleClotrimazoleVoriconazoleItraconazolePosaconazoleMiconazoleIsavuconazoleIsavuconazonium

Barbiturates (8)

PrimidonePhenobarbitalMethohexitalPentobarbitalButalbitalGlutethimideThiopentalSecobarbital

Benign prostatic hyperplasia (BPH) drugs (9)

TamsulosinFinasterideDoxazosinTerazosinAlfuzosinDutasterideTadalafilSilodosinTadalafil (PAH)

Benzodiazepines (18)

DiazepamLorazepamAlprazolamClonazepamMidazolamTemazepamChlordiazepoxideOxazepamClobazamClorazepateEstazolamFlurazepamQuazepamTriazolamRemimazolamAlprazolam XRFlunitrazepamLorazepam injection

Beta blockers (19)

PropranololMetoprololAtenololCarvedilolLabetalolBisoprololEsmololNadololAcebutololNebivololSotalolPindololCarteololBetaxololTimololCeliprololMetoprolol succinate ERPropranolol ERTalinolol

Beta-2 agonists (10)

AlbuterolLevalbuterolSalmeterolFormoterolArformoterolIndacaterolOlodaterolTerbutalineVilanterolAlbuterol nebulizer

Beta-lactam antibiotics (33)

AmoxicillinCephalexinCefdinirCefadroxilCefpodoximeCeftriaxoneErtapenemCefepimeMeropenemCefazolinDicloxacillinAmpicillinCeftazidimeCefiximePenicillin VAztreonamNafcillinOxacillinCefuroximeCloxacillinImipenemMethicillinCefotaximeCefoxitinCeftarolinePenicillin GPiperacillinCefaclorCefprozilCeftizoximeCephradineFlucloxacillinTicarcillin

Beta-lactamase inhibitors (6)

AvibactamClavulanateRelebactamSulbactamTazobactamVaborbactam

Biguanides (2)

MetforminMetformin ER

Bile acid sequestrants (3)

CholestyramineColesevelamColestipol

Bile acids (2)

UrsodiolObeticholic acid

Biologic disease-modifying antirheumatic drugs (DMARDs) (6)

AdalimumabEtanerceptInfliximabSarilumabTocilizumabRituximab

Bisphosphonates (5)

AlendronateIbandronateRisedronateZoledronic acidClodronate

Bleeding-associated medications (59)

WarfarinApixabanRivaroxabanDabigatranEdoxabanHeparinEnoxaparinFondaparinuxAspirinClopidogrelPrasugrelTicagrelorTiclopidineCilostazolDipyridamoleIbuprofenNaproxenDiclofenacIndomethacinKetorolacCelecoxibSertralineFluoxetineParoxetineCitalopramEscitalopramFluvoxamineVenlafaxineDuloxetineMeloxicamDonepezilMemantineNabumetoneRivastigmineEtodolacGalantamineSulindacPiroxicamTranexamic acidFlurbiprofenOxaprozinDiflunisalSalsalateKetoprofenMefenamic acidCapecitabineDeferasiroxFenoprofenIfosfamideMeclofenamateMifepristoneTolmetinDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchFluvoxamine CRMemantine XRParoxetine CRVenlafaxine XR

Bone and mineral metabolism drugs (17)

AlendronateIbandronateRaloxifeneDenosumabRisedronateCinacalcetCalcitonin (salmon)Sucroferric oxyhydroxideTeriparatideFerric citrateAbaloparatideParicalcitolZoledronic acidDoxercalciferolRomosozumabClodronatePalopeg­ teriparatide

Bone marrow suppression–associated medications (69)

MethotrexateAzathioprineCyclophosphamideCisplatinPaclitaxelVincristineLinezolidGanciclovirValganciclovirClozapineCarbamazepineFluorouracilHydroxyureaLenalidomideIbrutinibRuxolitinibPalbociclibImatinibVenetoclaxAcalabrutinibOsimertinibZanubrutinibAbemaciclibMercaptopurineEverolimusDasatinibSirolimusOlaparibFelbamateRibociclibNilotinibBosutinibTrametinibDabrafenibAlectinibNiraparibSotorasibRegorafenibErlotinibBexaroteneTucatinibLorlatinibCrizotinibVemurafenibMitotaneIdelalisibCeritinibCapecitabineVorinostatVandetanibTopotecanTemsirolimusRomidepsinBortezomibChloramphenicolDeferiproneDoxorubicinEtoposideIfosfamideIrinotecanProcainamideRibavirinTiclopidineTocainideCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRClozapine ODTClozapine oral suspension

Bone-loss–associated medications (34)

PrednisoneDexamethasoneHydrocortisoneMethyl­ prednisoloneBudesonidePhenytoinCarbamazepinePhenobarbitalPrimidoneValproic acidTopiramateHeparinOmeprazolePantoprazoleMedroxy­ progesteroneAnastrozoleLetrozoleExemestaneLeuprolidePioglitazoneDegarelixGoserelinPrednisoloneCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRDivalproex DRDivalproex ERDivalproex sprinkleHydrocortisone topicalMedroxyprogesterone depotTopiramate ERTopiramate ER (sprinkle)Valproate sodium IV

Bone-strengthening medications (14)

AlendronateRisedronateIbandronateZoledronic acidDenosumabTeriparatideAbaloparatideRomosozumabCalcitonin (salmon)RaloxifeneCholecalciferolErgocalciferolCalcitriolCalcium

Botanicals and herbal drugs (22)

BerberineSt John's wortApigeninBilobalideCurcuminGingerGinkgolide BGinkgotoxinHyperforinHypericinKaempferolLavenderMitragynineMyo-inositolPseudohypericinQuercetinRutinGinkgo biloba extractGreen teaL-TheanineSaffronSchisandra

Bowel-preparation drugs (4)

NeomycinBisacodylPEG 3350PEG 3350/ electrolytes

Bradycardia-associated medications (32)

MetoprololPropranololAtenololEsmololSotalolBisoprololCarvedilolLabetalolVerapamilDiltiazemDigoxinIvabradineAmiodaroneDronedaroneClonidineDonepezilRivastigmineGalantamineNeostigminePyridostigmineAdenosineDexmedetomidineNadololNebivololTimololClonidine ERClonidine ER suspensionDexmedetomidine sublingualDiltiazem ERMetoprolol succinate ERPropranolol ERVerapamil ER

Bradykinin receptor antagonists (1)

Icatibant

Bronchodilators (21)

AlbuterolTiotropiumIpratropiumUmeclidiniumEpinephrineLevalbuterolTheophyllineSalmeterolFormoterolArformoterolOlodaterolZileutonTerbutalineAminophyllineAclidiniumIndacaterolRevefenacinVilanterolAlbuterol nebulizerEnsifentrineIpratropium nasal

Calcimimetics (1)

Cinacalcet

Calcineurin inhibitors (6)

PimecrolimusCyclosporineTacrolimusVoclosporinCyclosporine ophthalmicTacrolimus ointment

Calcium channel blockers (CCBs) (15)

AmlodipineDiltiazemNifedipineVerapamilFelodipineNisoldipineIsradipineNicardipineNimodipineZiconotideClevidipineDiltiazem EREtripamilNifedipine ER (GITS)Verapamil ER

Cancer medications (112)

MethotrexateCyclosporineFluorouracilTacrolimusLeflunomideHydroxyureaMycophenolate mofetilAzathioprineLenalidomideAbirateroneEnzalutamideIbrutinibRuxolitinibTofacitinibUpadacitinibPalbociclibImatinibLeucovorinVenetoclaxAcalabrutinibApalutamideOsimertinibTeriflunomidePimecrolimusZanubrutinibAbemaciclibMercaptopurineEverolimusDasatinibSirolimusOlaparibRibociclibNilotinibBosutinibTrametinibDabrafenibAlectinibAprepitantNiraparibSotorasibGranisetronRegorafenibErlotinibBexaroteneCyclophosphamideTucatinibLorlatinibFilgrastimGivinostatCrizotinibPaclitaxelVemurafenibVoclosporinEliglustatMitotaneIdelalisibCisplatinRolapitantVincristineCeritinibCapecitabineVorinostatVandetanibTopotecanTemsirolimusRomidepsinNabiloneBelinostatGlucarpidaseIfosfamideNetupitantPanobinostatAbrocitinibAdalimumabBleomycinBortezomibConjugated estrogensDoxorubicinEstradiolEtanerceptEtoposideInfliximabIrinotecanNivolumabOspemifenePembrolizumabProcarbazineRituximabTamoxifenAfatinibAsciminibBevacizumabCapmatinibCyclosporine ophthalmicDacomitinibDarolutamideEstradiol transdermalEstradiol vaginalFruquintinibGefitinibPirtobrutinibPonatinibQuizartinibRipretinibRucaparibTacrolimus ointmentTemozolomideThalidomideToremifeneVepdegestrantVismodegibVorasidenib

Cannabinoids (7)

DronabinolCannabidiolNabilone2-Arachidonoyl­ glycerolAnandamideJWH-018Rimonabant

Carbapenems (3)

ErtapenemMeropenemImipenem

Carbonic anhydrase inhibitors (5)

DichlorphenamideAcetazolamideBrinzolamideDorzolamideMethazolamide

Cardiac glycosides (2)

DigoxinDigoxin immune Fab

Cardiovascular drugs (155)

AmlodipineLisinoprilLosartanMetoprololFurosemideApixabanHydrochloro­ thiazideCarvedilolClopidogrelDiclofenacEmpagliflozinSpironolactoneAtenololRivaroxabanDiltiazemHydralazineWarfarinIsosorbide mononitrateDapagliflozinValsartanPropranololNifedipineOlmesartanNaproxenAmiodaroneChlorthalidoneTorsemideNitroglycerinIrbesartanBenazeprilDoxazosinEnalaprilIcosapent ethylDigoxinDigoxin immune FabVerapamilRamiprilLidocaineNebivololPrazosinFlecainideRanolazineSotalolTelmisartanLabetalolBisoprololTicagrelorCilostazolDabigatranEnoxaparinIsosorbide dinitrateCandesartanMinoxidil oralIndapamideFelodipineFebuxostatPrasugrelDronedaroneDofetilidePropafenoneNadololEplerenoneGuanfacineFosinoprilDalfampridineAzilsartanMexiletineMacitentanCaptoprilAcebutololAmbrisentanQuinaprilTrandolaprilIvabradineTafamidisBaxdrostatHeparinRiociguatErtugliflozinVericiguatSelexipagTranexamic acidAliskirenPindololMoexiprilCarteololPerindoprilTreprostinilEthacrynic acidDipyridamoleFondaparinuxMavacamtenNisoldipineDisopyramideEdoxabanBosentanIsradipineNicardipineChloroquineQuinidineNimodipineSotagliflozinEpoprostenolDobutamineChlorothiazideZiconotideAjmalineAmyl nitriteAndexanet alfaAprindineAspirinCibenzolineClevidipineEncainideEprosartanEthacizineEtomidateGuanabenzHydroquinidineIbutilideIdarucizumabMethyldopaMoricizinePilsicainideProcainamideProtamine sulfateReserpineRosiglitazoneSacubitrilTiclopidineTocainideEXP3174 (E-3174)EXP3179MilrinoneNitroprussideAficamtenAprocitentanCeliprololDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchDiltiazem EREtripamilGuanfacine ERLidocaine injectionMetoprolol succinate ERMinoxidil topicalMoxonidineNifedipine ER (GITS)Omecamtiv mecarbilPropranolol ERRilmenidineSotaterceptTalinololVerapamil ER

Catechol-O-methyltransferase (COMT) inhibitors (3)

EntacaponeOpicaponeTolcapone

Central nervous system (CNS) depressants (172)

TramadolAlprazolamOxycodoneClonazepamLorazepamZolpidemDiazepamMorphineTemazepamLidocainePromethazinePrimidoneDoxepinNaloxoneFentanylHydromorphoneLoperamideDiphenoxylateEszopicloneMethadoneBuprenorphineSuzetriginePhenobarbitalNaltrexoneSuvorexantNaloxegolRamelteonZaleplonClobazamClorazepateBenzonatateTapentadolChlordiazepoxideTriazolamEstazolamMethylnaltrexoneDiphenhydramineHydrocodoneLemborexantOxymorphoneOxazepamEluxadolineDaridorexantMidazolamButorphanolNaldemedineCodeineFlumazenilPentazocineTasimelteonLevorphanolApomorphineMeperidineNalbuphineLofexidineDifenoxinBupivacaineTetracaineDexmedetomidineRopivacaineZiconotideFlurazepamKetamineMethohexitalNalmefenePentobarbitalQuazepamRemimazolamAlfentanilAlvimopanApigeninArticaineBeta-endorphinButalbitalCocaineDesfluraneDifelikefalinDynorphinEndomorphinsEnkephalinEthanolEthchlorvynolEtomidateGlutethimideHeroinIsofluraneMepivacaineMethaqualoneMitragynineNitrous oxideNociceptinO-desmethyl- tramadolOliceridineOrexin APhencyclidinePrilocaineProcainePropofolR-MethadoneRemifentanilS-MethadoneSalvinorin ASamidorphanSeltorexantSevofluraneSufentanilThiopentalTianeptineXylazineAllopregnanoloneAndrostanediolApalutamideBilobalideBrexanoloneCarisoprodolCefepimeCeftriaxoneCenobamateCiprofloxacinClarithromycinClozapineDHEASEnoxacinEnzalutamideErtapenemFelbamateGamma- Aminobutyric AcidGanaxoloneImipenemLevofloxacinMeprobamateMeropenemNorclobazamPenicillin VPicrotoxinPregnanoloneSecobarbitalStiripentolTaurineTHDOCTopiramateZincZuranoloneAlprazolam XRBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneClozapine ODTClozapine oral suspensionDexmedetomidine sublingualDoxepin low-dose (insomnia)FlunitrazepamHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERLidocaine injectionLorazepam injectionMorphine ER capsulesMorphine ER tabletsNaloxone nasal sprayNaltrexone ER injectionOxycodone CRPhenibutTopiramate ERTopiramate ER (sprinkle)Tramadol ERZolpidem CRZolpidem SLZolpidem SL middle-of-nightZolpidem oral spray

Cephalosporins (19)

CephalexinCefdinirCefadroxilCefpodoximeCeftriaxoneErtapenemCefepimeCefazolinCeftazidimeCefiximeAztreonamCefuroximeCefotaximeCefoxitinCeftarolineCefaclorCefprozilCeftizoximeCephradine

Cholesterol absorption inhibitors (1)

Ezetimibe

Cholinergic agonists (6)

AcetylcholineBethanecholPilocarpineCevimelineCarbacholXanomeline

Cholinesterase inhibitors (9)

PyridostigminePhysostigmineDonepezilRivastigmineGalantamineBenzgalantamineEdrophoniumNeostigmineSarin

Chronic interstitial nephropathy (6)

TacrolimusCyclosporineLithiumCyclosporine ophthalmicLithium ERTacrolimus ointment

Colony-stimulating factors (2)

FilgrastimPegfilgrastim

Combination medications (8)

ClavulanateCarbidopaCobicistatSacubitrilSamidorphanCarbidopa/ levodopaCarbidopa/ levodopa ERCarbidopa/ levodopa enteral

Constipation-associated medications (57)

MorphineOxycodoneHydrocodoneFentanylMethadoneBuprenorphineCodeineTramadolClozapineOlanzapineQuetiapineAmitriptylineImipramineClomipramineBenztropineOxybutyninTolterodineSolifenacinDarifenacinTrospiumVerapamilOndansetronErenumabCalciumRanolazineCalcium carbonateCholestyramineColesevelamColestipolDiltiazemDiphenhydramineDoxepinFerrous sulfateGranisetronHydroxyzine HClLanthanum carbonateNortriptylineSevelamerBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneClozapine ODTClozapine oral suspensionDiltiazem ERDoxepin low-dose (insomnia)Hydrocodone ER (q12h)Hydrocodone ER (q24h)Hydroxyzine IMMorphine ER capsulesMorphine ER tabletsOxybutynin EROxycodone CRQuetiapine XRTramadol ERVerapamil ER

Conventional disease-modifying antirheumatic drugs (DMARDs) (7)

MethotrexateHydroxy­ chloroquineSulfasalazineLeflunomideAzathioprineCyclosporineCyclosporine ophthalmic

Corticosteroids (30)

PrednisoneFluticasoneTriamcinoloneMethyl­ prednisolonePrednisoloneHydrocortisoneClobetasolTiotropiumIpratropiumDexamethasoneMometasoneUmeclidiniumBetamethasoneFluocinonideBudesonideFludrocortisoneFluorometholoneLoteprednolHalobetasolBeclomethasoneFlunisolideAclidiniumMifepristoneCiclesonideDes-ciclesonideFluticasone nasalHydrocortisone topicalIpratropium nasalTriamcinolone injectionVamorolone

Cough and cold medications (11)

GuaifenesinOlopatadineBenzonatateCetirizineDextromethorphanCodeineOxymetazolinePhenylephrinePseudoephedrineBrompheniramineChlorpheniramine

Crystal nephropathy (3)

AcyclovirMethotrexateValacyclovir

Cyclooxygenase (COX) inhibitors (29)

MeloxicamDiclofenacIbuprofenCelecoxibNaproxenKetorolacNabumetoneEtodolacIndomethacinSulindacPiroxicamFlurbiprofenOxaprozinDiflunisalSalsalateKetoprofenAcetaminophenMefenamic acidAspirinSalicylateBromfenacFenoprofenMeclofenamateTolmetin6-MNADiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchSulindac sulfide

Cytokine modulators (16)

AdalimumabEtanerceptInfliximabSarilumabTocilizumabSiltuximabDupilumabRuxolitinibTofacitinibUpadacitinibBimekizumabGuselkumabLebrikizumabMirikizumabOmalizumabTralokinumab

Cytotoxic chemotherapy (17)

ColchicineBleomycinCapecitabineCisplatinCyclophosphamideDoxorubicinEtoposideFluorouracilHydroxyureaIfosfamideIrinotecanMethotrexatePaclitaxelProcarbazineVincristinePhosphoramide mustardTemozolomide

DRESS-associated drugs (21)

AllopurinolCarbamazepineOxcarbazepinePhenytoinPhenobarbitalLamotrigineDapsoneVancomycinMinocyclineAbacavirNevirapineZonisamideCenobamateSulfamethoxazoleCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRLamotrigine XROxcarbazepine XRZiprasidoneZiprasidone IM

Decongestants (5)

OlopatadineCetirizineOxymetazolinePhenylephrinePseudoephedrine

Dementia medications (9)

DonepezilMemantineRivastigmineGalantamineBenzgalantamineBrexpiprazoleDonanemabLecanemabMemantine XR

Dermatologic drugs (26)

ClobetasolCalcitriolMometasoneBetamethasoneFluocinonideDupilumabMinoxidil oralTretinoinHalobetasolCalcipotrieneDapsoneIvermectinPimecrolimusAcitretinIsotretinoinTazaroteneCrisaboroleAlitretinoinBenzoyl peroxideChlorhexidineDeucravacitinibIxekizumabMinoxidil topicalRitlecitinibSecukinumabTirbanibulin

Diabetes medications (51)

MetforminInsulin glargineEmpagliflozinGlipizideGlimepirideDapagliflozinSitagliptinPioglitazoneInsulin lisproInsulin aspartInsulin detemirInsulin degludecLinagliptinRepaglinideCanagliflozinGlyburideAcarboseNateglinideSaxagliptinAlogliptinErtugliflozinBexagliflozinInsulin glulisinePramlintideSotagliflozinLixisenatideNPH insulinRegular insulinDulaglutideExenatideGlucagonLiraglutideOrforglipronRetatrutideRosiglitazoneSemaglutideTirzepatideTolbutamideGemigliptinGlipizide ERInsulin glargine U-300Insulin icodecLiraglutide (obesity)LobeglitazoneLuseogliflozinMetformin ERSemaglutide (obesity)Semaglutide oralSemaglutide oral (obesity)Tirzepatide (obesity)Voglibose

Dialyzable drugs (25)

LithiumValproic acidPhenobarbitalCarbamazepineGabapentinPregabalinLevetiracetamTopiramateMetforminAspirinTheophyllineSalicylateAcetaminophenAtenololCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRDivalproex DRDivalproex ERDivalproex sprinkleLithium ERMetformin ERTopiramate ERTopiramate ER (sprinkle)Valproate sodium IV

Dipeptidyl peptidase-4 (DPP-4) inhibitors (5)

SitagliptinLinagliptinSaxagliptinAlogliptinGemigliptin

Direct oral anticoagulants (DOACs) (5)

ApixabanRivaroxabanEdoxabanDabigatranBetrixaban

Direct renin inhibitors (1)

Aliskiren

Direct thrombin inhibitors (3)

DabigatranArgatrobanBivalirudin

Discontinued drugs (18)

NefazodoneCisaprideEncainideEthchlorvynolEzogabineGlutethimideLorcaserinMethaqualoneMethicillinMoricizinePhencyclidineRimonabantTegaserodTelithromycinTocainideSermorelinRanitidineTicarcillin

Disease-modifying antirheumatic drugs (DMARDs) (14)

MethotrexateSulfasalazineLeflunomidePenicillamineAdalimumabEtanerceptHydroxy­ chloroquineInfliximabRituximabSarilumabTocilizumabTofacitinibUpadacitinibBaricitinib

Disease-modifying multiple sclerosis drugs (11)

FingolimodDimethyl fumarateDiroximel fumarateTeriflunomideNatalizumabOfatumumabUblituximabOcrelizumabOzanimodPonesimodSiponimod

Diuretics (29)

FurosemideHydrochloro­ thiazideSpironolactoneChlorthalidoneTorsemideBumetanideDorzolamideMetolazoneIndapamideAcetazolamideSodium zirconium cyclosilicateFinerenoneEplerenoneBrinzolamideSucroferric oxyhydroxidePatiromerAmilorideFerric citrateLanthanum carbonateSodium polystyrene sulfonateMethazolamideSevelamerEthacrynic acidTriamtereneDichlorphenamideChlorothiazideMannitolGlycerinIsosorbide

Dopamine agonists (24)

PramipexoleRopiniroleRotigotineBromocriptineCabergolineApomorphineLevodopaAripiprazoleBrexpiprazoleCariprazineDehydro­ aripiprazoleDesmethyl­ cariprazineDidesmethyl­ cariprazineDopamineFenoldopamLysergic acid diethylamideNorclozapineAripiprazole lauroxil LAIAripiprazole lauroxil LAIAripiprazole monohydrate LAIAripiprazole monohydrate LAICarbidopa/ levodopaCarbidopa/ levodopa ERCarbidopa/ levodopa enteral

Dopamine antagonists (6)

MetoclopramideBuspironePromethazineTrimethobenzamideDomperidoneNorquetiapine

Dopamine reuptake inhibitors (33)

BupropionMethylphenidateModafinilArmodafinilDex­ methylphenidateSolriamfetolDesmethyl­ sertralineHydroxybupropionBenztropineCentanafadineCocaineLisdexamfetamineMethylenedioxy­ pyrovaleroneBupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERDexmethylphenidate XRMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patch

Dopamine-releasing agents (14)

AmphetamineAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)CathinoneDextroamphetamine IR tabletsDextroamphetamine oral solutionDextroamphetamine patchDextroamphetamine spansuleDextro­ amphetamineMephedroneMethamphetamineMixed amphetamine salts (triple-bead)Mixed amphetamine salts XR

Echinocandins (2)

MicafunginCaspofungin

Electrolyte replacements (10)

LinaclotideCalcium carbonateMg hydroxideMagnesium oxideMagnesium sulfatePotassium chlorideSodium bicarbonateCalcium chlorideCalcium gluconatePotassium citrate

Endocrine drugs (157)

LevothyroxineMetforminPrednisoneFluticasoneInsulin glargineEmpagliflozinSemaglutideGlipizideFinasterideTriamcinoloneMethyl­ prednisoloneDulaglutideGlimepirideDapagliflozinEstradiolSitagliptinPrednisolonePioglitazoneInsulin lisproInsulin aspartAmiodaroneHydrocortisoneClobetasolTiotropiumMelatoninInsulin detemirIpratropiumInsulin degludecTirzepatideAnastrozoleErgocalciferolLinagliptinDexamethasoneCalcitriolMometasoneTestosteroneUmeclidiniumDutasterideLiraglutideMethimazoleLetrozoleBetamethasoneFluocinonideLiothyronineBudesonideFludrocortisoneMegestrolMedroxy­ progesteroneResmetiromFluorometholoneRepaglinideLoteprednolCanagliflozinFinerenoneCinacalcetColesevelamBicalutamideGlucagonGlyburideHalobetasolExemestaneDesmopressinAcarboseBeclomethasoneNateglinideCalcipotrieneTeriparatideNorethindroneSaxagliptinAbaloparatideAlogliptinFlunisolideBromocriptinePropylthiouracilErtugliflozinElinzanetantLeuprolideCalcifediolSomatropinParicalcitolRibociclibExenatideBremelanotideOctreotideCrinecerfontTrametinibBexagliflozinDabrafenibAclidiniumInsulin glulisineDanazolMifepristoneCorticotropinLanreotideFezolinetantDrospirenoneClomipheneElagolixPramlintideDoxercalciferolLevonorgestrelSotagliflozinProgesteroneVandetanibAldosteroneConjugated estrogensDesogestrelDehydroepi­ androsteroneDHEASEthinyl estradiolGhrelinLeptinLixisenatideNorelgestrominNorgestimateNorgestrelNPH insulinOxytocinRegular insulinRetatrutideRosiglitazoneThyroid, desiccatedTolbutamideVasopressinAtosibanConivaptanNeuropeptide YOrforglipronSetmelanotideSubstance PTerlipressinTolvaptanBazedoxifeneEstradiol transdermalEstradiol vaginalEstriolEstroneEtonogestrelEtonogestrel implantFluticasone nasalGlipizide ERHydrocortisone topicalInsulin glargine U-300Ipratropium nasalLevonorgestrel IUDLiraglutide (obesity)Medroxyprogesterone depotMetformin ERPalopeg­ teriparatidePaltusotineSemaglutide (obesity)Semaglutide oralSemaglutide oral (obesity)Testosterone cypionateTirzepatide (obesity)Triamcinolone injectionUlipristal acetate

Endocrine therapies for cancer (11)

AnastrozoleLetrozoleTamoxifenAbirateroneBicalutamideExemestaneEnzalutamideApalutamideLeuprolideDegarelixGoserelin

Endogenous ligands (50)

2-Arachidonoyl­ glycerolATPAcetylcholineAdenosineAgmatineAldosteroneAllopregnanoloneAnandamideAndrostanediolAspartateBeta-endorphinBiocytinCoenzyme ACreatinineD-AlanineD-SerineDHEASDehydroepi­ androsteroneDopamineDynorphinEndomorphinsEnkephalinEpinephrineFADFMNGamma- Aminobutyric AcidGhrelinGlutamateGlycineHistamineKynurenic acidL-TheanineLeptinMelatoninNADNADPNeuropeptide YNitric oxideNociceptinNorepinephrineOrexin AOrexin BOxytocinPhenethylaminePregnenoloneSerotoninSubstance PTHDOCThiamine pyrophosphateVasopressin

Endothelin receptor antagonists (5)

MacitentanAmbrisentanBosentanSparsentanAprocitentan

Entry and fusion inhibitors (2)

MaravirocFostemsavir

Epidermal growth factor receptor (EGFR) inhibitors (5)

OsimertinibErlotinibAfatinibDacomitinibGefitinib

Erectile-dysfunction drugs (6)

SildenafilTadalafilAvanafilVardenafilYohimbineTadalafil (PAH)

Ergot alkaloids (5)

BromocriptineDihydro­ ergotamineErgotamineCabergolineMethylergonovine

Erythropoiesis-stimulating agents (ESAs) (2)

Darbepoetin alfaEpoetin alfa

Estrogens (13)

EstradiolAnastrozoleRaloxifeneTamoxifenOspemifeneClomipheneConjugated estrogensEndoxifenEthinyl estradiolEstradiol transdermalEstradiol vaginalEstriolEstrone

Expectorants/mucolytics (3)

GuaifenesinN-acetylcysteine (NAC)Acetylcysteine

Extrapyramidal symptom (EPS)–associated medications (41)

HaloperidolFluphenazineTrifluoperazinePerphenazineChlorpromazineThiothixeneLoxapineRisperidonePaliperidoneAmisulprideOlanzapineAripiprazoleBrexpiprazoleCariprazineMetoclopramideProchlorperazinePromethazineDroperidolAmoxapineAsenapineIloperidoneLurasidoneMolindonePimozideThioridazineTrimethobenzamideZiprasidoneAripiprazole lauroxil LAIAripiprazole lauroxil LAIAripiprazole monohydrate LAIAripiprazole monohydrate LAIAsenapine transdermalFluphenazine decanoate LAIHaloperidol decanoate LAIHaloperidol injectionLoxapine inhaledPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIZiprasidone IM

Fall-risk medications (146)

MidazolamDexmedetomidineKetamineMethohexitalPentobarbitalRemimazolamTrazodoneQuetiapineMirtazapineZolpidemCyclobenzaprineTizanidineHydroxyzine HClOlanzapineAmitriptylineMeclizineTemazepamPromethazinePrimidoneDoxepinClozapineFentanylEszopiclonePhenobarbitalCarisoprodolSuvorexantChlorpromazineCyproheptadineRamelteonLumateperoneTriazolamEstazolamLemborexantDaridorexantThioridazineTasimelteonTrimipramineDoxylamineFlurazepamQuazepamGabapentinTramadolAlprazolamOxycodoneClonazepamLorazepamBuspironePregabalinBaclofenRisperidoneClonidineDiazepamMorphineMethocarbamolNortriptylineHydromorphoneProchlorperazinePaliperidoneMethadoneBuprenorphineBrexpiprazoleScopolamineImipramineZaleplonClobazamClorazepateClomipramineTapentadolDronabinolChlordiazepoxideCenobamateAsenapineLoxapineMetaxaloneChlorzoxazonePerampanelOrphenadrineHydrocodoneIloperidoneOxymorphoneOxazepamGabapentin enacarbilButorphanolCodeinePentazocineLevorphanolMeprobamateApomorphineMeperidineNalbuphineAcetaminophenZiconotideNabiloneAlfuzosinDiphenhydramineDonepezilDoxazosinFurosemideGuanfacineHaloperidolHydrochloro­ thiazideMemantineMethyldopaMidodrineOxybutyninPrazosinSecobarbitalTamsulosinTerazosinAlprazolam XRAsenapine transdermalBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneClonidine ERClonidine ER suspensionClozapine ODTClozapine oral suspensionDexmedetomidine sublingualDoxepin low-dose (insomnia)Guanfacine ERHaloperidol decanoate LAIHaloperidol injectionHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERHydroxyzine IMLorazepam injectionLoxapine inhaledMemantine XRMorphine ER capsulesMorphine ER tabletsOxybutynin EROxycodone CRPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIQuetiapine XRTramadol ERZolpidem CRZolpidem SLZolpidem SL middle-of-nightZolpidem oral spray

Fertility drugs (3)

DanazolClomipheneLetrozole

Fibrates (2)

FenofibrateGemfibrozil

Fibrinolytics (2)

AlteplaseTenecteplase

First-generation antihistamines (11)

DiphenhydramineDimenhydrinateDoxylamineChlorpheniramineBrompheniramineHydroxyzine HClMeclizinePromethazineCyproheptadineKetotifenHydroxyzine IM

First-generation antipsychotics (17)

HaloperidolChlorpromazineFluphenazinePerphenazineTrifluoperazineThioridazineThiothixeneLoxapineMolindonePimozideProchlorperazineDroperidolFlupentixolFluphenazine decanoate LAIHaloperidol decanoate LAIHaloperidol injectionLoxapine inhaled

Fluoroquinolones (11)

CiprofloxacinLevofloxacinOfloxacinMoxifloxacinEnoxacinDelafloxacinGatifloxacinGemifloxacinNemonoxacinNorfloxacinSparfloxacin

Folate antagonists (4)

MethotrexatePyrimethamineTrimethoprimSulfamethoxazole

Gabapentinoids (3)

GabapentinPregabalinGabapentin enacarbil

Gastrointestinal drugs (71)

OmeprazolePantoprazoleFamotidineOndansetronEsomeprazoleMeclizineSucralfateLactulosePromethazineLansoprazoleMetoclopramideDexlansoprazoleNaloxoneLoperamideDiphenoxylateProchlorperazineUrsodiolLubiprostoneNaloxegolRabeprazolePlecanatideUpadacitinibCimetidineDronabinolMisoprostolPrucaloprideMethylnaltrexoneEluxadolineHyoscyamineNaldemedineTenapanorObeticholic acidAlosetronAprepitantGranisetronNizatidineDifenoxinRolapitantDoxylamineTrimethobenzamideMannitolAmisulprideNabiloneBisacodylDomperidoneMg hydroxidePEG 3350SennaCalcium carbonateCisaprideCromolynDocusateLinaclotideMagnesium oxideNetupitantPsylliumSimethiconeSodium bicarbonateTegaserodAcacia gumAl/Mg antacidAluminum hydroxideBismuth subsalicylateCalcium polycarbophilInulinMethylcelluloseNaloxone nasal sprayPEG 3350/ electrolytesRanitidineVonoprazanWheat dextrin

General anesthetics (9)

PropofolEtomidateKetamineThiopentalMethohexitalSevofluraneIsofluraneDesfluraneNitrous oxide

Genitourinary drugs (25)

TamsulosinFinasterideOxybutyninMirabegronDoxazosinTerazosinSolifenacinAlfuzosinSildenafilDutasterideTolterodineVibegronTrospiumTadalafilSilodosinFesoterodineDarifenacinAvanafilVardenafilYohimbineBethanecholPentosan polysulfatePhenazopyridineOxybutynin ERTadalafil (PAH)

Glucagon (1)

Glucagon

Glucagon-like peptide-1 (GLP-1) receptor agonists (13)

SemaglutideLiraglutideDulaglutideExenatideLixisenatideTirzepatideOrforglipronRetatrutideLiraglutide (obesity)Semaglutide (obesity)Semaglutide oralSemaglutide oral (obesity)Tirzepatide (obesity)

Glucocorticoids (24)

PrednisoneTriamcinoloneMethyl­ prednisolonePrednisoloneDexamethasoneMifepristoneBeclomethasoneBetamethasoneBudesonideCiclesonideClobetasolFlunisolideFluocinonideFluorometholoneFluticasoneHalobetasolHydrocortisoneLoteprednolMometasoneDes-ciclesonideFluticasone nasalHydrocortisone topicalTriamcinolone injectionVamorolone

Glycopeptide antibiotics (1)

Vancomycin

Gonadotropin-releasing hormone (GnRH) agonists and antagonists (4)

LeuprolideElagolixDegarelixGoserelin

Gout medications (6)

AllopurinolColchicineFebuxostatProbenecidLesinuradRasburicase

Hair-loss–associated medications (35)

Valproic acidLithiumTopiramateLamotrigineCarbamazepineHeparinWarfarinPropranololMetoprololLevothyroxineMethimazoleIsotretinoinAcitretinLeuprolideAnastrozoleLetrozoleMethotrexateCyclophosphamideDutasterideFinasterideMinoxidil oralCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRDivalproex DRDivalproex ERDivalproex sprinkleLamotrigine XRLithium ERMetoprolol succinate ERMinoxidil topicalPropranolol ERTopiramate ERTopiramate ER (sprinkle)Valproate sodium IV

Hematologic drugs (37)

ApixabanClopidogrelRivaroxabanWarfarinTicagrelorCilostazolDabigatranEnoxaparinPrasugrelFerric citrateTafamidisHeparinTranexamic acidFelbamateDipyridamoleFondaparinuxEdoxabanAndexanet alfaAspirinChloramphenicolIdarucizumabProtamine sulfateTiclopidineDarbepoetin alfaEpoetin alfaFerrous sulfateArgatrobanAvatrombopagBetrixabanBivalirudinClopidogrel active metaboliteEltrombopagPegfilgrastimProthrombin complex concentrate (4-factor)RoxadustatVadadustatVoxelotor

Hematopoietic drugs (6)

FilgrastimDarbepoetin alfaEpoetin alfaAvatrombopagEltrombopagPegfilgrastim

Hemodynamic renal effects (reversible) (38)

IbuprofenNaproxenDiclofenacIndomethacinKetorolacLisinoprilLosartanFurosemideMeloxicamCelecoxibValsartanOlmesartanIrbesartanBenazeprilBumetanideEnalaprilRamiprilTelmisartanNabumetoneEtodolacFosinoprilSulindacAzilsartanCaptoprilQuinaprilTrandolaprilPiroxicamMoexiprilPerindoprilFlurbiprofenOxaprozinDiflunisalSalsalateKetoprofenMefenamic acidDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patch

Hemostatic drugs (9)

Tranexamic acidAlteplaseAndexanet alfaDesmopressinIdarucizumabPhytonadioneProtamine sulfateTenecteplaseProthrombin complex concentrate (4-factor)

Hepatitis antivirals (19)

EntecavirTenofovirLamivudineDasabuvirGlecaprevirLedipasvirOmbitasvirParitaprevirPibrentasvirVelpatasvirAdefovirPeginterferon alfaRibavirinBemnifosbuvirDaclatasvirElbasvirGrazoprevirSimeprevirSofosbuvir

Hepatobiliary drugs (8)

UrsodiolRifaximinNeomycinObeticholic acidLactuloseResmetiromElafibranorSeladelpar

Hepatotoxic medications (51)

AtorvastatinRosuvastatinSimvastatinPravastatinEzetimibeKetoconazoleFluconazoleLovastatinMethotrexateIcosapent ethylFenofibrateMethimazoleGemfibrozilAzathioprinePitavastatinNiacinRifampinFerric citrateBempedoic acidPropylthiouracilFluvastatinVoriconazoleIsoniazidItraconazolePosaconazoleFelbamateIsavuconazoniumMicafunginGriseofulvinNefazodoneAcetaminophenAmiodaroneBosentanDantroleneEntecavirFezolinetantIdelalisibLeflunomideMaravirocNevirapineRegorafenibSparsentanTerbinafineTeriflunomideTolcaponeTolvaptanValproic acidDivalproex DRDivalproex ERDivalproex sprinkleValproate sodium IV

Herpesvirus antivirals (10)

ValacyclovirAcyclovirFamciclovirValganciclovirGanciclovirLetermovirCidofovirFoscarnetMaribavirPenciclovir

Histamine H2 receptor antagonists (5)

FamotidineCimetidineNizatidineHistamineRanitidine

Hormonal cancer therapies (14)

AnastrozoleLetrozoleRaloxifeneTamoxifenAbirateroneBicalutamideExemestaneEnzalutamideApalutamideLeuprolideOspemifeneDegarelixGoserelinToremifene

Hormonal contraceptives (15)

MegestrolMedroxy­ progesteroneNorethindroneDrospirenoneLevonorgestrelDesogestrelEthinyl estradiolNorelgestrominNorgestimateNorgestrelEtonogestrelEtonogestrel implantLevonorgestrel IUDMedroxyprogesterone depotUlipristal acetate

Hormone replacement therapy (12)

EstradiolConjugated estrogensProgesteroneTestosteroneLevothyroxineLiothyronineFludrocortisoneHydrocortisoneEstradiol transdermalEstradiol vaginalHydrocortisone topicalTestosterone cypionate

Human immunodeficiency virus (HIV) antiretrovirals (27)

LamivudineDoravirineEtravirineAbacavirMaravirocRilpivirineFostemsavirCabotegravirElvitegravirAtazanavirBictegravirCobicistatDarunavirDolutegravirEfavirenzEmtricitabineLenacapavirLopinavirNevirapineRaltegravirRitonavirTenofovirDidanosineIslatravirLenacapavir (PrEP)Tenofovir alafenamideZidovudine

Huntington disease medications (2)

DeutetrabenazineTetrabenazine

Hydroxymethylglutaryl-CoA (HMG-CoA) reductase inhibitors (8)

AtorvastatinRosuvastatinSimvastatinPravastatinLovastatinGemfibrozilPitavastatinFluvastatin

Hyperglycemia-associated medications (28)

PrednisoneDexamethasoneHydrocortisoneOlanzapineClozapineQuetiapineRisperidoneTacrolimusCyclosporineSirolimusEverolimusNiacinHydrochloro­ thiazideChlorthalidonePhenytoinSomatropinTriamcinoloneMethyl­ prednisoloneBudesonideFludrocortisonePrednisoloneClozapine ODTClozapine oral suspensionCyclosporine ophthalmicHydrocortisone topicalQuetiapine XRTacrolimus ointmentTriamcinolone injection

Hypertension-associated medications (86)

AmphetamineMethamphetamineMethylphenidateLisdexamfetaminePhenterminePseudoephedrinePhenylephrineEpinephrineNorepinephrineDopamineMidodrineBupropionVenlafaxineDuloxetineDesvenlafaxineTranylcyprominePhenelzineSelegilineMeloxicamDiclofenacIbuprofenCelecoxibNaproxenCyclosporineKetorolacNaloxoneNabumetoneTacrolimusEtodolacIndomethacinSulindacDextro­ amphetaminePiroxicamDextromethorphanFlurbiprofenOxaprozinDiflunisalSalsalateKetoprofenIsocarboxazidMefenamic acidAtomoxetineDarbepoetin alfaEpoetin alfaErenumabLevomilnacipranMirabegronPhendimetrazinePrednisoneSolriamfetolAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)Bupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERCyclosporine ophthalmicDextroamphetamine IR tabletsDextroamphetamine oral solutionDextroamphetamine patchDextroamphetamine spansuleDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchMixed amphetamine salts (triple-bead)Mixed amphetamine salts XRNaloxone nasal spraySelegiline transdermalTacrolimus ointmentVenlafaxine XR

Hypoglycemia-associated medications (39)

GlipizideGlyburideGlimepirideTolbutamideRepaglinideNateglinideSemaglutideLiraglutideDulaglutideExenatideTirzepatideAcarboseMetforminInsulin glargineDapagliflozinSitagliptinPioglitazoneInsulin lisproInsulin aspartInsulin detemirInsulin degludecLinagliptinSaxagliptinAlogliptinErtugliflozinBexagliflozinInsulin glulisinePramlintideSotagliflozinNPH insulinRegular insulinGlipizide ERInsulin glargine U-300Liraglutide (obesity)Metformin ERSemaglutide (obesity)Semaglutide oralSemaglutide oral (obesity)Tirzepatide (obesity)

Hyponatremia-associated medications (40)

Hydrochloro­ thiazideChlorthalidoneIndapamideSertralineFluoxetineParoxetineCitalopramEscitalopramVenlafaxineDuloxetineCarbamazepineOxcarbazepineEslicarbazepineDesmopressinClozapineRisperidoneHaloperidolCyclophosphamideVincristineMilnacipranLevomilnacipranGepironeZuranoloneChlorothiazideAmitriptylineMetolazoneMirtazapineOxytocinCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRClozapine ODTClozapine oral suspensionFluvoxamineFluvoxamine CRHaloperidol decanoate LAIHaloperidol injectionOxcarbazepine XRParoxetine CRVenlafaxine XR

Hypotension-associated medications (63)

PrazosinDoxazosinTerazosinTamsulosinClonidineGuanfacineLisinoprilLosartanAmlodipineVerapamilDiltiazemNitroglycerinHydralazineMinoxidil oralSildenafilTadalafilClozapineQuetiapineChlorpromazineTrazodoneAmitriptylineMetoprololCarvedilolAtenololPropranololNifedipineNebivololLabetalolBisoprololFelodipineNadololPhenytoinAcebutololPindololCarteololNisoldipineIsradipineNicardipineChloroquineNimodipineMethohexitalRemimazolamAlfuzosinAvanafilIloperidoneIsosorbide dinitrateIsosorbide mononitrateMethyldopaSilodosinVardenafilClonidine ERClonidine ER suspensionClozapine ODTClozapine oral suspensionDiltiazem ERGuanfacine ERMetoprolol succinate ERMinoxidil topicalNifedipine ER (GITS)Propranolol ERQuetiapine XRTadalafil (PAH)Verapamil ER

Immune checkpoint inhibitors (2)

NivolumabPembrolizumab

Immunomodulators (50)

CyclosporineAdalimumabTacrolimusLeflunomideMycophenolate mofetilAzathioprineEtanerceptLenalidomideApremilastTofacitinibUpadacitinibDimethyl fumarateTocilizumabTeriflunomidePirfenidoneFingolimodSarilumabInfliximabDiroximel fumarateVoclosporinAbrocitinibBimekizumabGuselkumabIcatibantLebrikizumabLinvoseltamabMirikizumabOfatumumabOmalizumabPacritinibTralokinumabUblituximabAnifrolumabBaricitinibBelimumabCyclosporine ophthalmicDeucravacitinibEfgartigimodEtrasimodIxekizumabOzanimodPonesimodRemibrutinibRisankizumabRitlecitinibSecukinumabSiponimodTacrolimus ointmentThalidomideUstekinumab

Immunosuppressants (29)

PrednisoneCyclosporineAdalimumabTacrolimusLeflunomideMycophenolate mofetilAzathioprineEtanerceptLenalidomideApremilastTofacitinibUpadacitinibDimethyl fumarateTocilizumabTeriflunomidePirfenidoneEverolimusSirolimusFingolimodSarilumabInfliximabDiroximel fumarateCyclophosphamideVoclosporinAbrocitinibMifepristoneRituximabCyclosporine ophthalmicTacrolimus ointment

Inflammatory bowel disease (IBD) drugs (15)

AdalimumabMesalamineSulfasalazineTofacitinibUpadacitinibBalsalazideInfliximabAzathioprineBudesonideMercaptopurineMethotrexateMirikizumabEtrasimodMesalamine DROzanimod

Influenza antivirals (4)

AmantadineBaloxavir marboxilOseltamivirAmantadine ER

Inhaled antimuscarinics (6)

AclidiniumGlycopyrrolateIpratropiumRevefenacinTiotropiumUmeclidinium

Inhaled corticosteroids (12)

FluticasoneTiotropiumIpratropiumMometasoneUmeclidiniumCiclesonideBeclomethasoneFlunisolideAclidiniumBudesonideTriamcinoloneDes-ciclesonide

Inhaled medications (28)

FluticasoneTiotropiumIpratropiumMometasoneUmeclidiniumBudesonideTobramycinBeclomethasoneLoxapineFlunisolideAclidiniumAmyl nitriteDesfluraneIsofluraneNitric oxideSevofluraneAlbuterolArformoterolCiclesonideCromolynFormoterolIndacaterolLevalbuterolOlodaterolRevefenacinSalmeterolVilanterolEnsifentrine

Inotropes (10)

MidodrineDroxidopaItraconazoleDobutamineDigoxinDopamineEpinephrineIsoproterenolMilrinoneOmecamtiv mecarbil

Insulins (29)

Insulin glargineEmpagliflozinGlipizideGlimepirideDapagliflozinSitagliptinPioglitazoneInsulin lisproInsulin aspartInsulin detemirInsulin degludecLinagliptinRepaglinideCanagliflozinGlyburideAcarboseSaxagliptinAlogliptinErtugliflozinBexagliflozinInsulin glulisinePramlintideSotagliflozinLixisenatideNPH insulinRegular insulinGlipizide ERInsulin glargine U-300Insulin icodec

Integrase strand-transfer inhibitors (INSTIs) (5)

RaltegravirDolutegravirBictegravirElvitegravirCabotegravir

Intensive-care medications (41)

LorazepamAmiodaroneMidodrineSotalolPermethrinMexiletineDroxidopaDisopyramideIdelalisibDobutamineDexmedetomidinePentobarbitalRemimazolamAtracuriumCisatracuriumCurareEncainideIfosfamideMetocurineMivacuriumMoricizineNorepinephrinePancuroniumPropofolRocuroniumSt John's wortSuccinylcholineTocainideVasopressinVecuroniumAlteplaseClevidipineEpinephrineEsmololFentanylMidazolamMilrinoneNicardipineNitroprussideDexmedetomidine sublingualLorazepam injection

Interferons (1)

Peginterferon alfa

Interleukin inhibitors (15)

SarilumabTocilizumabSiltuximabDupilumabBimekizumabGuselkumabLebrikizumabMirikizumabTralokinumabBenralizumabIxekizumabMepolizumabRisankizumabSecukinumabUstekinumab

Intranasal medications (18)

FluticasoneTriamcinoloneAzelastineMometasoneBeclomethasoneAmilorideEsketamineButorphanolDihydro­ ergotamineZavegepantCiclesonideFlunisolideBudesonideDesmopressinNaloxoneOxymetazolineSumatriptanEtripamil

Intravenous fluids (4)

LinaclotideIV lipid emulsionMannitolSodium bicarbonate

Iron preparations (3)

Sucroferric oxyhydroxideFerric citrateFerrous sulfate

Janus kinase (JAK) inhibitors (11)

TofacitinibAbrocitinibPacritinibRuxolitinibUpadacitinibBaricitinibFedratinibFostamatinibMomelotinibPeficitinibRitlecitinib

Kinase inhibitors (49)

AcalabrutinibAlectinibBosutinibCeritinibCrizotinibDasatinibErlotinibIbrutinibImatinibLorlatinibNilotinibOsimertinibRegorafenibTucatinibVandetanibZanubrutinibNetarsudilAbemaciclibAbrocitinibDabrafenibIdelalisibPacritinibPalbociclibRibociclibRuxolitinibSotorasibTofacitinibTrametinibUpadacitinibVemurafenibAfatinibAsciminibBaricitinibCapmatinibDacomitinibDeucravacitinibFedratinibFostamatinibFruquintinibGefitinibMomelotinibNintedanibPeficitinibPirtobrutinibPonatinibQuizartinibRemibrutinibRipretinibRitlecitinib

Labor and delivery drugs (12)

CabergolineBromocriptineFezolinetantTerbutalineAtosibanOxytocinBetamethasoneDinoprostoneMagnesium sulfateMethylergonovineMisoprostolCarboprost

Laxatives (26)

LactuloseNaloxoneLubiprostoneNaloxegolPlecanatidePrucaloprideMethylnaltrexoneNaldemedineTenapanorMannitolBisacodylMg hydroxidePEG 3350SennaDocusateGlycerinLinaclotideMagnesium oxidePsylliumAcacia gumCalcium polycarbophilInulinMethylcelluloseNaloxone nasal sprayPEG 3350/ electrolytesWheat dextrin

Leukotriene modifiers (3)

MontelukastZafirlukastZileuton

Lincosamides (1)

Clindamycin

Lipid-lowering drugs (29)

AtorvastatinRosuvastatinSimvastatinPravastatinEzetimibeLovastatinIcosapent ethylFenofibrateEvolocumabGemfibrozilAlirocumabCholestyramineColestipolPitavastatinColesevelamNiacinBempedoic acidFluvastatinBerberineLactuloseObeticholic acidOmega-3 fatty acidsPancrelipasePentosan polysulfateSucralfateUrsodiolEnlicitideInclisiranLerodalcibep

Lipopeptide antibiotics (1)

Daptomycin

Lithium salts (2)

LithiumLithium ER

Local anesthetics (10)

LidocaineBupivacaineRopivacaineMepivacainePrilocaineProcaineTetracaineArticaineCocaineLidocaine injection

Long-acting injectables (LAIs) (22)

CabotegravirDegarelixGoserelinLeuprolideAripiprazole lauroxil LAIAripiprazole lauroxil LAIAripiprazole monohydrate LAIAripiprazole monohydrate LAIFluphenazine decanoate LAIHaloperidol decanoate LAIMedroxyprogesterone depotNaltrexone ER injectionOlanzapine pamoate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIRisperidone LAIRisperidone LAIRisperidone LAIRisperidone LAIRisperidone LAI

Loop diuretics (4)

FurosemideTorsemideBumetanideEthacrynic acid

Luminal (nonsystemic gastrointestinal) agents (24)

PhenobarbitalEluxadolineCholestyramineColesevelamColestipolFidaxomicinLanthanum carbonateNeomycinNystatinPatiromerRifaximinSevelamerSodium zirconium cyclosilicateSucralfateVancomycinAcacia gumAl/Mg antacidAluminum hydroxideBismuth subsalicylateCalcium polycarbophilInulinMethylcelluloseSodium butyrateWheat dextrin

Macrolides (4)

AzithromycinErythromycinClarithromycinTelithromycin

Mast cell stabilizers (3)

CromolynKetotifenOlopatadine

Mechanistic target of rapamycin (mTOR) inhibitors (3)

EverolimusSirolimusTemsirolimus

Meglitinides (2)

RepaglinideNateglinide

Menopause medications (9)

ElinzanetantFezolinetantConjugated estrogensEstradiolOspemifeneProgesteroneBazedoxifeneEstradiol transdermalEstradiol vaginal

Metabolites (79)

(Desmethyl-) mirtazapine1-PP4-ene-VPA5-HMT5-hydroxy­ tryptophan6-MNA7-OH loxapine7-OHmitragynine7-amino­ clonazepam7-amino­ flunitrazepam8-OH-AmoxapineAcetylcholineAcroleinAllopregnanoloneAmoxapineBenazeprilatCalcifediolCalcitriolChloroacet­ aldehydeClopidogrel active metaboliteDehydro­ aripiprazoleDes-ciclesonideDesglymidodrineDesipramineDesmethyl­ cariprazineDesmethyl­ clomipramineDesmethyl­ sertralineDesvenlafaxineDextrorphanDidesmethyl­ cariprazineDopamineEXP3174 (E-3174)EXP3179EnalaprilatEndoxifenFluorouracilFosinoprilatGabapentinHydroxybupropionHydroxy­ nefazodoneL-MethylfolateLatanoprost free acidMesalamineMethylcobalaminMilsaperidoneMorphineMorphine-3glucuronideMorphine-6glucuronideNAPQINorclobazamNorclozapineNordiazepamNordoxepinNorelgestrominNorepinephrineNorfluoxetineNoribogaineNormeperidineNorquetiapineNortriptylineO-desmethyl- tramadolPaliperidonePenciclovirPerindoprilatPhenobarbitalPhosphoramide mustardPsilocinPyridoxal-5'- phosphateQuinaprilatRamiprilatSerotoninSirolimusSulindac sulfideTemsavirTetrahydro­cannabinolTrandolaprilatmCPPα-hydroxy­ alprazolamα-methyl­ norepinephrine

Methylphenidates (18)

MethylphenidateDex­ methylphenidateDexmethylphenidate XRMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchSerdexmethylphenidate

Microtubule inhibitors (4)

ColchicinePaclitaxelVincristineTirbanibulin

Mineralocorticoid receptor antagonists (MRAs) (3)

FinerenoneEplerenoneSpironolactone

Mineralocorticoids (4)

DexamethasoneFludrocortisoneEplerenoneAldosterone

Monoamine oxidase B (MAO-B) inhibitors (4)

SelegilineRasagilineSafinamideSelegiline transdermal

Monoamine oxidase inhibitors (MAOIs) (6)

PhenelzineTranylcypromineIsocarboxazidSelegilineMoclobemideSelegiline transdermal

Monobactams (1)

Aztreonam

Monoclonal antibodies (47)

EvolocumabAdalimumabAlirocumabDupilumabDenosumabTocilizumabSarilumabInfliximabErenumabFremanezumabGalcanezumabIdarucizumabRomosozumabSiltuximabBimekizumabFilgrastimGuselkumabLebrikizumabMirikizumabNatalizumabNivolumabOfatumumabOmalizumabPegvisomantPembrolizumabRituximabTralokinumabUblituximabVutrisiranAfliberceptAnifrolumabBelimumabBenralizumabBevacizumabDonanemabEfgartigimodFaricimabIxekizumabLecanemabMepolizumabNirsevimabOcrelizumabRanibizumabRisankizumabSecukinumabTezepelumabUstekinumab

Mood stabilizers (30)

LithiumValproic acidLamotrigineCarbamazepineAripiprazoleAsenapineCariprazineLurasidoneOlanzapineOxcarbazepineQuetiapineRisperidoneZiprasidoneAripiprazole lauroxil LAIAripiprazole lauroxil LAIAripiprazole monohydrate LAIAripiprazole monohydrate LAIAsenapine transdermalCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRDivalproex DRDivalproex ERDivalproex sprinkleLamotrigine XRLithium EROxcarbazepine XRQuetiapine XRValproate sodium IVZiprasidone IM

Mucosal protective agents (2)

SucralfateMisoprostol

Multiple sclerosis (MS) drugs (13)

DalfampridineDimethyl fumarateTeriflunomideFingolimodDiroximel fumarateCorticotropinNatalizumabOfatumumabUblituximabOcrelizumabOzanimodPonesimodSiponimod

Muscarinic agonists (8)

BethanecholPilocarpineCevimelineCarbacholXanomelineAcetylcholineAceclidineNorclozapine

Muscle relaxants (10)

CyclobenzaprineTizanidineBaclofenMethocarbamolCarisoprodolMetaxaloneChlorzoxazoneOrphenadrineDantroleneBotulinum toxin

Myopathy/rhabdomyolysis-associated medications (17)

AtorvastatinSimvastatinRosuvastatinPravastatinLovastatinFluvastatinPitavastatinGemfibrozilFenofibrateColchicineDaptomycinHydroxy­ chloroquineRaltegravirEzetimibeIcosapent ethylNiacinBempedoic acid

Narrow therapeutic index (NTI) drugs (240)

LithiumWarfarinDigoxinTheophyllinePhenytoinCarbamazepineValproic acidTacrolimusCyclosporineSirolimusEverolimusVancomycinGentamicinTobramycinAmikacinLevothyroxineMethotrexateAbemaciclibAcitretinAjmalineAlfentanilAlprazolamAminophyllineAmitriptylineAmoxapineAmphotericin BApixabanAprindineAtracuriumAzathioprineBosutinibBotulinum toxinBumetanideBuprenorphineCalcitriolCapecitabineCarbacholChloroquineCibenzolineCisaprideCisatracuriumCisplatinCitalopramClomipramineClonazepamClozapineCodeineColchicineCrizotinibCurareCyclophosphamideDabigatranDabrafenibDalfampridineDantroleneDasatinibDeferoxamineDesfluraneDesipramineDesmethyl­ clomipramineDiazepamDigoxin immune FabDihydro­ ergotamineDimercaprolDisopyramideDizocilpineDobutamineDomoic acidDomperidoneDoxepinDroperidolEdetate calcium disodiumEdoxabanEncainideEpoprostenolErgotamineEthacizineEthacrynic acidEthchlorvynolEthosuximideEtomidateFelbamateFenoldopamFentanylFingolimodFlecainideFlibanserinFluorouracilFondaparinuxFoscarnetFosphenytoinGanciclovirGlutethimideHaloperidolHeparinHeroinHexamethoniumHydrocodoneHydromorphoneHydroquinidineIbrutinibIbutilideIfosfamideImipramineInsulin aspartInsulin degludecInsulin detemirInsulin glargineInsulin glulisineInsulin lisproIsocarboxazidIsofluraneIsoproterenolKainateKetorolacLamotrigineLeflunomideLenalidomideLevorphanolLiothyronineLorazepamMaprotilineMecamylamineMefloquineMeperidineMeprobamateMercaptopurineMethadoneMethaqualoneMethohexitalMethsuximideMetocurineMexiletineMitotaneMivacuriumMoricizineMorphineMycophenolate mofetilNeostigmineNilotinibNiraparibNitroprussideNordoxepinNortriptylineNPH insulinOlaparibOsimertinibOxycodoneOxymorphonePaclitaxelPalbociclibPancuroniumPentamidinePentobarbitalPhenelzinePhenoxybenzaminePhentolaminePhysostigminePicrotoxinPilsicainidePimozidePolymyxin BPotassium chloridePralidoximePrimidoneProcainamideProcarbazineProtamine sulfateProtriptylineR-MethadoneRegadenosonRegorafenibRegular insulinRemifentanilRibociclibRivaroxabanRuxolitinibS-MethadoneSarinSevofluraneSotalolStrychnineSufentanilTamoxifenTapentadolTemsirolimusTeriflunomideThiopentalThioridazineThyroid, desiccatedTocainideTofacitinibTolcaponeTopotecanTrametinibTranylcypromineTriazolamTrimipramineTucatinibUpadacitinibValganciclovirVandetanibVecuroniumVemurafenibVenetoclaxVincristineVoclosporinVoriconazoleXylazineZiconotideAlprazolam XRBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRClozapine ODTClozapine oral suspensionCyclosporine ophthalmicDivalproex DRDivalproex ERDivalproex sprinkleDoxepin low-dose (insomnia)Haloperidol decanoate LAIHaloperidol injectionHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERInsulin glargine U-300Lamotrigine XRLithium ERLorazepam injectionMorphine ER capsulesMorphine ER tabletsOxycodone CRTacrolimus ointmentValproate sodium IV

Nasal corticosteroids (6)

FluticasoneBeclomethasoneBudesonideFlunisolideMometasoneTriamcinolone

Neuraminidase inhibitors (1)

Oseltamivir

Neuroleptic malignant syndrome (NMS)–associated medications (2)

MetoclopramidePromethazine

Neurology medications (111)

GabapentinClonazepamDonepezilPregabalinMemantineLevetiracetamLamotriginePropranololRopiniroleTopiramateBenztropineSumatriptanPramipexoleCarbamazepinePrimidoneOxcarbazepineLacosamideRizatriptanAmantadineCandesartanPhenobarbitalZonisamideRivastigmineRimegepantGalantamineUbrogepantTrihexyphenidylDeutetrabenazineClobazamRasagilineEntacaponePhenytoinDalfampridineBrivaracetamAtogepantNaratriptanDimethyl fumarateEslicarbazepineCenobamateMexiletineRotigotineTeriflunomideEletriptanPerampanelZolmitriptanSelegilineCannabidiolFingolimodGabapentin enacarbilRufinamideTetrabenazineFelbamateDihydro­ ergotamineIstradefyllineCarbidopaTiagabineOpicaponeDiroximel fumarateEthosuximideLasmiditanLevodopaFrovatriptanCorticotropinAlmotriptanZavegepantMethsuximideVigabatrinFenfluramineStiripentolTolcaponeFosphenytoinGanaxoloneErgotaminePentobarbitalBotulinum toxinCapsaicinErenumabFremanezumabGalcanezumabValproic acidAmifampridineEdaravoneEzogabineKynurenic acidLevocarnitineRiluzoleAmantadine ERCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRCarbidopa/ levodopaCarbidopa/ levodopa ERCarbidopa/ levodopa enteralDivalproex DRDivalproex ERDivalproex sprinkleDonanemabEfgartigimodLacosamide ERLamotrigine XRLecanemabMemantine XROmaveloxoloneOxcarbazepine XRPropranolol ERSelegiline transdermalSumatriptan SC injectionSumatriptan nasalTopiramate ERTopiramate ER (sprinkle)Valproate sodium IV

Neuromuscular blockers (9)

AtracuriumCisatracuriumCurareMetocurineMivacuriumPancuroniumRocuroniumSuccinylcholineVecuronium

Neurotransmitters (24)

2-Arachidonoyl­ glycerolATPAcetylcholineAdenosineAnandamideAspartateBeta-endorphinDopamineDynorphinEnkephalinEpinephrineGHB (Oxybate)Gamma- Aminobutyric AcidGlutamateGlycineHistamineMixed-salt oxybatesNeuropeptide YNociceptinNorepinephrineOrexin AOrexin BSerotoninSubstance P

Neutropenia-associated medications (21)

ClozapineCarbamazepineMethimazolePropylthiouracilDeferiproneDapsoneLinezolidGanciclovirValganciclovirMethotrexateAzathioprineCyclophosphamideColchicineRituximabTiclopidineVancomycinCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRClozapine ODTClozapine oral suspension

Nicotinic agonists (9)

Nicotine gumAcetylcholineVareniclineSuccinylcholineCarbacholNicotine inhalerNicotine lozengeNicotine nasal sprayNicotine patch

Nicotinic antagonists (10)

MecamylamineHexamethoniumRocuroniumVecuroniumPancuroniumAtracuriumCisatracuriumCurareMetocurineMivacurium

Nitrates (4)

Isosorbide mononitrateNitroglycerinIsosorbide dinitrateAmyl nitrite

Nitroimidazoles (1)

Metronidazole

Non-drug (17)

AMPAApple juiceCreatinineDizocilpineDomoic acidEthylene glycolGrapefruit juiceKainateMethanolMilkN-methylD-aspartateOrange juicePicrotoxinPolycyclic Aromatic HydrocarbonsSarinStrychnineTyramine

Non-nucleoside reverse transcriptase inhibitors (NNRTIs) (5)

DoravirineEtravirineRilpivirineEfavirenzNevirapine

Nonbenzodiazepine hypnotics (7)

ZolpidemEszopicloneZaleplonZolpidem CRZolpidem SLZolpidem SL middle-of-nightZolpidem oral spray

Nonopioid analgesics (38)

MeloxicamDiclofenacIbuprofenCelecoxibNaproxenKetorolacLidocaineNabumetoneBromfenacEtodolacIndomethacinSulindacMisoprostolPiroxicamFlurbiprofenOxaprozinDiflunisalSalsalateKetoprofenAcetaminophenMefenamic acidBupivacaineTetracaineRopivacaineArticaineAspirinCocaineMepivacaineN-acetylcysteine (NAC)PrilocaineProcaineSalicylateCapsaicinSuzetrigineDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchLidocaine injection

Nonsteroidal anti-inflammatory drugs (NSAIDs) (29)

MeloxicamDiclofenacIbuprofenCelecoxibNaproxenKetorolacNabumetoneBromfenacEtodolacIndomethacinSulindacMisoprostolPiroxicamFlurbiprofenOxaprozinDiflunisalSalsalateKetoprofenMefenamic acidAspirinSalicylateFenoprofenMeclofenamateTolmetin6-MNADiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchSulindac sulfide

Norepinephrine reuptake inhibitors (NRIs) (62)

SertralineTramadolDuloxetineBupropionFluoxetineVenlafaxineParoxetineDoxepinMethylphenidateAtomoxetineClomipramineMilnacipranLevomilnacipranViloxazineProtriptylineAmoxapine8-OH-AmoxapineDesmethyl­ clomipramineDesmethyl­ sertralineHydroxybupropionNordoxepinNorfluoxetineNorquetiapineAmitriptylineCentanafadineCocaineDesipramineDesvenlafaxineDex­ methylphenidateImipramineLisdexamfetamineMaprotilineMethylenedioxy­ pyrovaleroneNortriptylineReboxetineTapentadolZiprasidoneBupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERDexmethylphenidate XRDoxepin low-dose (insomnia)Methylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchParoxetine CRTramadol ERVenlafaxine XRZiprasidone IM

Norepinephrine-releasing agents (13)

AmphetamineAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)CathinoneMethamphetamineMethylenedioxy­ methamphetamineMixed amphetamine salts (triple-bead)Mixed amphetamine salts XRPhendimetrazinePhenterminePseudoephedrineTyramine

Norepinephrine–dopamine reuptake inhibitors (NDRIs) (25)

BupropionCentanafadineDex­ methylphenidateMethylphenidateSolriamfetolBupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERDexmethylphenidate XRMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patch

Nucleoside and nucleotide reverse transcriptase inhibitors (NRTIs) (5)

LamivudineAbacavirEmtricitabineEntecavirTenofovir

Omega-3 fatty acids (2)

Icosapent ethylOmega-3 fatty acids

Oncology drugs (109)

MethotrexateCyclosporineAnastrozoleLetrozoleRaloxifeneFluorouracilTacrolimusLeflunomideHydroxyureaMycophenolate mofetilMegestrolAzathioprineTamoxifenLenalidomideAbirateroneBicalutamideExemestaneEnzalutamideIbrutinibRuxolitinibTofacitinibUpadacitinibPalbociclibImatinibLeucovorinVenetoclaxAcalabrutinibApalutamideOsimertinibTeriflunomidePimecrolimusZanubrutinibAbemaciclibMercaptopurineEverolimusDasatinibSirolimusOlaparibLeuprolideRibociclibNilotinibBosutinibTrametinibDabrafenibAlectinibNiraparibSotorasibRegorafenibErlotinibBexaroteneCyclophosphamideTucatinibLorlatinibGivinostatCrizotinibPaclitaxelVemurafenibVoclosporinEliglustatMitotaneIdelalisibCisplatinVincristineCeritinibCapecitabineVorinostatVandetanibTopotecanTemsirolimusRomidepsinBelinostatGlucarpidaseIfosfamideLorcaserinPanobinostatBleomycinBortezomibDoxorubicinEtoposideIrinotecanNivolumabPembrolizumabProcarbazineRituximabAfatinibAsciminibBevacizumabCapmatinibCyclosporine ophthalmicDacomitinibDarolutamideDexrazoxaneFruquintinibGefitinibMesnaNintedanibPirtobrutinibPonatinibQuizartinibRasburicaseRipretinibRucaparibTacrolimus ointmentTemozolomideThalidomideToremifeneVepdegestrantVismodegibVorasidenib

Ophthalmic drugs (41)

LatanoprostClonidinePrednisoloneAzelastineTimololBrimonidineBimatoprostLidocaineOfloxacinDorzolamideKetotifenTravoprostLifitegrastOlopatadineScopolamineNetarsudilFluorometholoneLoteprednolBromfenacAcetazolamidePilocarpineBrinzolamideAtropineMethazolamideCetirizineBetaxololCyclopentolateCarteololFlurbiprofenOxymetazolinePhenylephrinePolymyxin BTropicamideTetracaineMannitolAceclidineCarbacholAcoltremonAfliberceptFaricimabRanibizumab

Opioid agonists (28)

MorphineOxycodoneHydrocodoneHydromorphoneOxymorphoneFentanylAlfentanilSufentanilRemifentanilMethadoneCodeineMeperidineTramadolTapentadolLevorphanolOliceridineDifelikefalinDifenoxinDiphenoxylateHeroinLoperamideHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERMorphine ER capsulesMorphine ER tabletsOxycodone CRTramadol ER

Opioid antagonists (10)

NaloxoneNaltrexoneNalmefeneNaloxegolNaldemedineMethylnaltrexoneAlvimopanSamidorphanNaloxone nasal sprayNaltrexone ER injection

Opioid partial agonists (9)

BuprenorphineButorphanolNalbuphinePentazocineBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxone

Opioid use disorder (OUD) medications (13)

MethadoneBuprenorphineNaltrexoneNPH insulinLofexidineNaloxoneBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneNaloxone nasal sprayNaltrexone ER injection

Opioids (59)

MorphineOxycodoneHydrocodoneHydromorphoneOxymorphoneFentanylAlfentanilSufentanilRemifentanilMethadoneCodeineMeperidineTramadolTapentadolLevorphanolOliceridineBuprenorphineButorphanolNalbuphinePentazocineDifelikefalinAlvimopanBeta-endorphinDifenoxinDiphenoxylateDynorphinEluxadolineEndomorphinsEnkephalinHeroinLoperamideMethylnaltrexoneMitragynineNaldemedineNalmefeneNaloxegolNaloxoneNaltrexoneNociceptinO-desmethyl- tramadolR-MethadoneS-MethadoneSalvinorin ASamidorphanTianeptineBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERMorphine ER capsulesMorphine ER tabletsNaloxone nasal sprayNaltrexone ER injectionOxycodone CRTramadol ER

Orphan drugs (26)

AcoramidisAmifampridineEdaravoneGivinostatIcatibantIvacaftorLumacaftorPegvisomantRiluzoleSetmelanotideTafamidisTrofinetideVutrisiranLevocarnitineEliglustatAficamtenCrinecerfontOmaveloxoloneSeladelparSepiapterinSodium benzoateSotaterceptTezacaftorVamoroloneVatiquinoneVoxelotor

Orthostatic hypotension–associated medications (31)

PrazosinDoxazosinTerazosinTamsulosinClozapineQuetiapineChlorpromazineTrazodoneAmitriptylineImipramineLevodopaRopinirolePramipexoleSildenafilTadalafilClonidineAlfuzosinCarvedilolDoxepinFurosemideIloperidoneLabetalolMethyldopaNortriptylineClonidine ERClonidine ER suspensionClozapine ODTClozapine oral suspensionDoxepin low-dose (insomnia)Quetiapine XRTadalafil (PAH)

Osmotic diuretics (3)

MannitolGlycerinIsosorbide

Osteoclast inhibitors (7)

DenosumabAlendronateRisedronateIbandronateZoledronic acidCalcitonin (salmon)Clodronate

Osteoporosis medications (13)

AlendronateIbandronateRaloxifeneDenosumabRisedronateCalcitonin (salmon)TeriparatideAbaloparatideZoledronic acidRomosozumabCalcium carbonateCholecalciferolClodronate

Otic drugs (6)

CefdinirOfloxacinPolymyxin BCefuroximeClavulanateNeomycin

Over-the-counter (OTC) medications (44)

OmeprazoleIbuprofenMelatoninClotrimazoleLoperamideGuaifenesinDiphenhydraminePhenazopyridineCannabidiolCetirizineNicotine gumDextromethorphanDoxylamineAcetaminophen5-hydroxy­ tryptophanAspirinBisacodylCaffeineCalcium carbonateCholecalciferolDimenhydrinateDocusateGingerLoratadineMg hydroxideNorgestrelOmega-3 fatty acidsPEG 3350SennaSimethiconeZincα-TocopherolBerberineCurcuminFerrous sulfateMagnesium oxideMyo-inositolNicotinamidePregnenolonePsylliumQuercetinSarcosineTryptophanL-Theanine

Overactive bladder drugs (10)

OxybutyninMirabegronSolifenacinTolterodineVibegronTrospiumFesoterodineDarifenacin5-HMTOxybutynin ER

Oxazolidinones (2)

LinezolidTedizolid

Pain medications (132)

GabapentinTramadolDuloxetineMeloxicamOxycodoneDiclofenacIbuprofenPregabalinCelecoxibNaproxenMorphineMethocarbamolSumatriptanKetorolacLidocaineNaloxoneFentanylHydromorphoneLoperamideDiphenoxylateRizatriptanNabumetoneMethadoneBuprenorphineSuzetrigineNaltrexoneRimegepantSuvorexantBromfenacNaloxegolEtodolacIndomethacinUbrogepantSulindacAtogepantTapentadolMisoprostolNaratriptanMexiletineMetaxaloneEletriptanOrphenadrineMethylnaltrexonePiroxicamZolmitriptanHydrocodonePentosan polysulfateLemborexantPhenazopyridineOxymorphoneEluxadolineDaridorexantButorphanolNaldemedineDihydro­ ergotamineFlurbiprofenOxaprozinCodeineLasmiditanDiflunisalFrovatriptanAlmotriptanPentazocineSalsalateLevorphanolApomorphineKetoprofenElagolixZavegepantMeperidineNalbuphineLofexidineDifenoxinAcetaminophenMefenamic acidBupivacaineTetracaineErgotamineRopivacaineZiconotideNalmefeneAlfentanilAlvimopanArticaineAspirinBeta-endorphinCapsaicinCocaineDifelikefalinDynorphinEndomorphinsEnkephalinHeroinIV lipid emulsionMepivacaineMitragynineNociceptinO-desmethyl- tramadolOliceridineOrexin APrilocaineProcaineR-MethadoneRemifentanilS-MethadoneSalicylateSalvinorin ASamidorphanSeltorexantSubstance PSufentanilTianeptineBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERLidocaine injectionMorphine ER capsulesMorphine ER tabletsNaloxone nasal sprayNaltrexone ER injectionOxycodone CRSumatriptan SC injectionSumatriptan nasalTramadol ER

Pancreatic enzyme replacements (1)

Pancrelipase

Parathyroid hormone (PTH) analogs (3)

TeriparatideAbaloparatidePalopeg­ teriparatide

Parkinson disease medications (22)

RopiniroleBenztropinePramipexoleAmantadineTrihexyphenidylRasagilinePimavanserinEntacaponeRotigotineSelegilineIstradefyllineCarbidopaOpicaponeLevodopaTolcaponeApomorphineSafinamideAmantadine ERCarbidopa/ levodopaCarbidopa/ levodopa ERCarbidopa/ levodopa enteralSelegiline transdermal

Penicillins (13)

AmoxicillinDicloxacillinAmpicillinPenicillin VAztreonamNafcillinOxacillinCloxacillinMethicillinPenicillin GPiperacillinFlucloxacillinTicarcillin

Peripherally acting mu-opioid receptor antagonists (PAMORAs) (4)

NaloxegolNaldemedineMethylnaltrexoneAlvimopan

Phosphate binders (5)

Sucroferric oxyhydroxideFerric citrateCalcium carbonateLanthanum carbonateSevelamer

Phosphodiesterase (PDE) inhibitors (17)

SildenafilTadalafilAvanafilVardenafilCilostazolPentoxifyllineRoflumilastTheophyllineApremilastDipyridamoleCrisaboroleAminophyllineCaffeineMilrinoneEnsifentrineNerandomilastTadalafil (PAH)

Phosphodiesterase-5 (PDE5) inhibitors (5)

SildenafilTadalafilAvanafilVardenafilTadalafil (PAH)

Pituitary and hypothalamic drugs (18)

DesmopressinLeuprolideSomatropinOctreotideCorticotropinLanreotideElagolixGhrelinOrexin ABromocriptineCabergolineCrinecerfontDegarelixGoserelinPegvisomantSermorelinVasopressinPaltusotine

Poisoning agents (5)

Domoic acidEthylene glycolMethanolPicrotoxinStrychnine

Polyene antifungals (2)

NystatinAmphotericin B

Polymyxin antibiotics (1)

Polymyxin B

Potassium binders (3)

PatiromerSodium zirconium cyclosilicateSodium polystyrene sulfonate

Potassium-elevating medications (23)

SpironolactoneEplerenoneFinerenoneAmilorideTriamtereneLisinoprilEnalaprilRamiprilLosartanValsartanIrbesartanOlmesartanAliskirenTrimethoprimHeparinTacrolimusCyclosporineBenazeprilCandesartanSulfamethoxazoleTelmisartanCyclosporine ophthalmicTacrolimus ointment

Potassium-lowering medications (19)

FurosemideBumetanideTorsemideEthacrynic acidHydrochloro­ thiazideChlorthalidoneIndapamideMetolazoneAlbuterolLevalbuterolPatiromerSodium zirconium cyclosilicateSodium polystyrene sulfonateAmphotericin BChlorothiazideInsulin lisproSodium bicarbonateTerbutalineAlbuterol nebulizer

Potassium-sparing diuretics (5)

AmilorideTriamtereneEplerenoneFinerenoneSpironolactone

Prodrugs (37)

PrednisoneClopidogrelLatanoprostValacyclovirEnalaprilMidodrinePrimidoneNabumetoneCefpodoximeLisdexamfetamineTamoxifenCyanocobalaminCiclesonideFesoterodineSulindacClorazepateFamciclovirBalsalazideValganciclovirDroxidopaGabapentin enacarbilIsavuconazoniumCodeineIsotretinoinFostemsavirDoxercalciferolCapecitabineFosphenytoinBenzgalantamineHeroinMethyldopaPsilocybinCyclophosphamideIfosfamideLumacaftorTramadolTramadol ER

Progestins (14)

MegestrolMedroxy­ progesteroneNorethindroneDrospirenoneLevonorgestrelProgesteroneDesogestrelNorelgestrominNorgestimateNorgestrelEtonogestrelEtonogestrel implantLevonorgestrel IUDMedroxyprogesterone depot

Prokinetic drugs (8)

ErythromycinMetoclopramidePrucaloprideHyoscyamineAlosetronCisaprideDomperidoneTegaserod

Proprotein convertase subtilisin/kexin type 9 (PCSK9) inhibitors (5)

AlirocumabEvolocumabEnlicitideInclisiranLerodalcibep

Protease inhibitors (10)

DarunavirRitonavirAtazanavirNelfinavirGlecaprevirIndinavirLopinavirNirmatrelvirParitaprevirSaquinavir

Proteasome inhibitors (1)

Bortezomib

Proton pump inhibitors (PPIs) (6)

OmeprazoleEsomeprazoleLansoprazoleDexlansoprazolePantoprazoleRabeprazole

Pulmonary hypertension drugs (13)

SildenafilTadalafilMacitentanAmbrisentanRiociguatSelexipagTreprostinilBosentanEpoprostenolNitric oxideVericiguatSotaterceptTadalafil (PAH)

Purinergic receptor modulators (10)

ClopidogrelTicagrelorPrasugrelATPTiclopidineAdenosineCaffeineDipyridamoleIstradefyllineRegadenoson

QT-prolonging medications (163)

SotalolDofetilideThioridazineNilotinibDisopyramidePimozideQuinidineVandetanibDroperidolAzithromycinDonepezilCitalopramCiprofloxacinOndansetronFluconazoleAmiodaroneLevofloxacinHydroxy­ chloroquineErythromycinMoxifloxacinHaloperidolCilostazolMethadoneDronedaroneChlorpromazineClarithromycinOsimertinibIvabradineRibociclibChloroquinePentamidineEscitalopramTizanidineVenlafaxinePromethazineOfloxacinNortriptylineFlecainideRanolazineAlfuzosinTolterodineProchlorperazineZiprasidonePaliperidoneFluorouracilTacrolimusRivastigmineTamoxifenBicalutamidePerphenazineImipraminePimavanserinImatinibApalutamideDesipramineIloperidoneDasatinibVoriconazoleFingolimodPosaconazoleLeuprolideGepironeTetrabenazineFelbamateRilpivirineMilsaperidoneBosutinibEfavirenzDabrafenibPitolisantMifepristoneGranisetronIsradipineApomorphineGivinostatCrizotinibVemurafenibVoclosporinEliglustatTrimipramineLofexidineCeritinibCapecitabineVorinostatRomidepsinAmisulprideRemimazolam8-OH-AmoxapineAjmalineAmitriptylineAmoxapineAsenapineCibenzolineCisaprideClomipramineClozapineDesmethyl­ clomipramineDolasetronDomperidoneDoxepinHydroquinidineHydroxyzine HClIbutilideLoperamideLoxapineMaprotilinemCPPNorclozapineNordoxepinNorquetiapineOlanzapinePanobinostatProcainamideProtriptylineQuetiapineR-MethadoneS-MethadoneSulpirideTrazodoneTrifluoperazineRisperidoneBuprenorphinePropafenoneFluphenazineThiothixeneVardenafilMolindone7-OH loxapineAsenapine transdermalBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneClozapine ODTClozapine oral suspensionDoxepin low-dose (insomnia)EndoxifenFluphenazine decanoate LAIHaloperidol decanoate LAIHaloperidol injectionHydroxyzine IMHydroxyzine pamoateLapatinibLoxapine inhaledNAPAOlanzapine pamoate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPazopanibPralsetinibQuetiapine XRRisperidone LAIRisperidone LAIRisperidone LAIRisperidone LAIRisperidone LAISorafenibTacrolimus ointmentVenlafaxine XRZiprasidone IM

QT-shortening medications (5)

CenobamateRufinamideDigoxinIsavuconazoleIsavuconazonium

Raises creatinine without kidney injury (5)

BictegravirCimetidineCobicistatDolutegravirTrimethoprim

Renal and electrolyte drugs (61)

FurosemideHydrochloro­ thiazideEmpagliflozinSpironolactoneGlipizideChlorthalidoneTorsemideHydrocortisoneIrbesartanLinaclotideBumetanideKetorolacLinagliptinCalcitriolDorzolamideMetolazoneFludrocortisoneIndapamideAcetazolamideSodium zirconium cyclosilicateFinerenoneNadololEplerenoneFosinoprilBrinzolamideSucroferric oxyhydroxidePatiromerAmilorideFerric citrateProbenecidLanthanum carbonateAcamprosateSodium polystyrene sulfonateMethazolamideErtugliflozinSevelamerEthacrynic acidDemeclocyclineTriamtereneCorticotropinNitrofurantoinDichlorphenamideChlorothiazideMannitolAmphotericin BTemsirolimusEtomidateFenoldopamTerlipressinVasopressinYohimbineCinacalcetConivaptanParicalcitolPotassium chlorideTolvaptanCalcium chlorideCalcium gluconateGlipizide ERHydrocortisone topicalPotassium citrate

Renally cleared drugs (225)

LisinoprilGabapentinMetforminHydrochloro­ thiazideFamotidineAmoxicillinAlendronateCephalexinPregabalinAtenololMemantineBaclofenCiprofloxacinLevetiracetamSitagliptinValsartanClonidineFluconazoleTopiramateOlmesartanValacyclovirChlorthalidoneLevofloxacinMethotrexateTiotropiumLevocetirizineCefdinirAcyclovirDoxycyclinePramipexoleDigoxinDigoxin immune FabOfloxacinMidodrineSotalolDorzolamideFolic acidIbandronateMethenamine hippuratePaliperidoneMetolazoneVareniclineEnoxaparinAmantadineHydroxyureaTrospiumCandesartanCefadroxilCefpodoximeGentamicinVancomycinOlopatadineLenalidomideCeftriaxoneAcetazolamideDofetilideCyanocobalaminNadololRisedronatePyridostigmineTobramycinGlycopyrrolateBrinzolamideTrimethoprimErtapenemDaptomycinEntecavirCimetidineDalfampridineAmilorideFosfomycinCefepimeLeucovorinNaratriptanMeropenemPrucaloprideTenofovirCefazolinCaptoprilAlogliptinEthambutolNeomycinAcamprosatePhenazopyridineLamivudineLevocarnitineCetirizineTranexamic acidDicloxacillinAmpicillinCarteololGanciclovirCarbidopaSolriamfetolCeftazidimeCefiximeExenatideBremelanotideFondaparinuxAmikacinMethenamine mandelateEdoxabanEmtricitabinePenicillin VAztreonamZoledronic acidNitrofurantoinDeferiproneNizatidinePramlintideVigabatrinPhenterminePenicillamineTrientineDichlorphenamideCisplatinTrofinetideDeferoxaminePolymyxin BTrimethobenzamideChlorothiazideThiamineTopotecanMannitolCefuroximeCidofovirPentamidineSuccimerAmphotericin BCycloserineLithiumAmisulprideClavulanateAndexanet alfaAscorbic acidCarbacholCibenzolineClodronateDifelikefalinDimercaprolEdetate calcium disodiumEdrophoniumEprosartanFexofenadineGlucarpidaseHydroxocobalaminIdarucizumabImipenemIV lipid emulsionMecamylamineMethicillinMethyldopaMetocurinePancuroniumPilsicainidePralidoximeProtamine sulfatePseudoephedrinePyridoxineRegadenosonRocuroniumSodium thiosulfateSugammadexSulpirideTeriflunomidePentosan polysulfate1-PPAcoltremonAcoramidisActivated charcoalAMPACalciumCefotaximeCefoxitinCeftarolineCurareDiazoxideDomoic acidEnoxacinFenoprofenFlucytosineFoscarnetHexamethoniumIsosorbideKainateKynurenic acidLanthanum carbonateLeptinMagnesiumMg hydroxideMagnesium sulfateMeclofenamateN-methylD-aspartatePatiromerPenicillin GPiperacillinPEG 3350Potassium chloridePrussian blueRevefenacinSevelamerSodium bicarbonateSodium zirconium cyclosilicateSodium polystyrene sulfonateTolmetinZincAmantadine ERBaricitinibClonidine ERClonidine ER suspensionDesglymidodrineEnalaprilatGlycopyrrolate inhaledL-TheanineLithium ERMemantine XRMetformin ERPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPenciclovirTicarcillinTopiramate ERTopiramate ER (sprinkle)

Renin–angiotensin–aldosterone system (RAAS) inhibitors (31)

LisinoprilMontelukastCiprofloxacinBenazeprilEnalaprilRamiprilPromethazineFosinoprilTofacitinibCaptoprilQuinaprilTrandolaprilLevocarnitineAliskirenMoexiprilPerindoprilTolcaponeDroperidolRomosozumabAzilsartanCandesartanEprosartanEXP3174 (E-3174)EXP3179IrbesartanLosartanOlmesartanSacubitrilTelmisartanValsartanEnalaprilat

Respiratory drugs (68)

AlbuterolFluticasoneMontelukastAmoxicillinLevofloxacinTiotropiumCefdinirIpratropiumMometasoneMoxifloxacinUmeclidiniumSildenafilGuaifenesinBudesonideEpinephrineDupilumabCefpodoximeRoflumilastTadalafilLevalbuterolTobramycinCiclesonideTheophyllineBeclomethasoneBenzonatateCromolynMacitentanEthambutolSalmeterolZafirlukastLoxapineAmbrisentanPirfenidoneFlunisolideRiociguatSelexipagTreprostinilFormoterolArformoterolOlodaterolAclidiniumZileutonBosentanTerbutalineNalbuphineEpoprostenolCefuroximeDexmedetomidineAminophyllineAmyl nitriteIndacaterolNitric oxideSevofluraneVilanterolAcetylcysteineAlbuterol nebulizerBenralizumabDexmedetomidine sublingualEnsifentrineFluticasone nasalIpratropium nasalLoxapine inhaledMepolizumabNerandomilastNintedanibTadalafil (PAH)TezacaftorTezepelumab

Respiratory-depressant medications (60)

MorphineOxycodoneHydrocodoneFentanylMethadoneBuprenorphineCodeineTramadolAlprazolamLorazepamDiazepamClonazepamMidazolamTemazepamPhenobarbitalPentobarbitalPropofolEtomidateKetamineGabapentinPregabalinZolpidemEszopicloneCarisoprodolBaclofenAlfentanilButorphanolDifenoxinDiphenoxylateHeroinHydromorphoneLevorphanolMeperidineNalbuphineOliceridineOxymorphonePentazocinePromethazineQuazepamRemifentanilSufentanilTapentadolAlprazolam XRBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERLorazepam injectionMorphine ER capsulesMorphine ER tabletsOxycodone CRTramadol ERZolpidem CRZolpidem SLZolpidem SL middle-of-nightZolpidem oral spray

Retinoids (6)

TretinoinAcitretinIsotretinoinTazaroteneBexaroteneAlitretinoin

Reversal agents (20)

NaloxoneCyproheptadineDantroleneDextromethorphanDeferasiroxFlumazenilDeferiproneDeferoxamineNalmefenePhysostigmineN-acetylcysteine (NAC)PhytonadioneAndexanet alfaDigoxin immune FabGlucarpidaseIdarucizumabProtamine sulfateSugammadexNaloxone nasal sprayProthrombin complex concentrate (4-factor)

Reverse transcriptase inhibitors (11)

AbacavirDoravirineEfavirenzEmtricitabineEntecavirEtravirineLamivudineNevirapineRilpivirineTenofovirAdefovir

Rifamycins (4)

RifampinRifabutinRifapentineRifaximin

Risk Evaluation and Mitigation Strategy (REMS) medications (25)

IsotretinoinMifepristoneLenalidomideVigabatrinEsketamineRiociguatBosentanAcitretinAlosetronAlvimopanAmbrisentanBuprenorphineDofetilideFelbamateMacitentanMethadoneMycophenolate mofetilSotalolSparsentanFentanylBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxone

Schedule I controlled substances (15)

HeroinLysergic acid diethylamidePsilocybinPsilocinN,N-dimethyl­ tryptamineMescalineMethylenedioxy­ methamphetamineJWH-018CathinoneIbogaineMethylenedioxy­ pyrovaleroneMephedroneMethaqualoneSalvinorin ADizocilpine

Schedule II controlled substances (59)

AmphetamineDextro­ amphetamineMethamphetamineLisdexamfetamineDex­ methylphenidateCocaineMorphineOxycodoneHydrocodoneHydromorphoneOxymorphoneFentanylMethadoneMeperidineTapentadolCodeinePentobarbitalAlfentanilLevorphanolMethylphenidateNabiloneOliceridineRemifentanilSecobarbitalSufentanilAmobarbitalAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)Dexmethylphenidate XRDextroamphetamine IR tabletsDextroamphetamine oral solutionDextroamphetamine patchDextroamphetamine spansuleGlutethimideHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchMixed amphetamine salts (triple-bead)Mixed amphetamine salts XRMorphine ER capsulesMorphine ER tabletsOxycodone CRR-MethadoneS-Methadone

Schedule III controlled substances (14)

BuprenorphineKetamineDronabinolTestosteroneButalbitalPhendimetrazineBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneButabarbitalDanazolEsketamine

Schedule IV controlled substances (48)

AlprazolamLorazepamDiazepamClonazepamChlordiazepoxideOxazepamTemazepamTriazolamMidazolamClobazamClorazepateEstazolamFlurazepamQuazepamZolpidemEszopicloneZaleplonSuvorexantLemborexantDaridorexantModafinilArmodafinilTramadolCarisoprodolPhentermineButorphanolPentazocineDifenoxinRemimazolamSolriamfetolAlprazolam XRBrexanoloneEluxadolineHalazepamLorazepam injectionLorcaserinMeprobamateMethohexitalPhenobarbitalPrimidoneStiripentolThiopentalTramadol ERZolpidem CRZolpidem SLZolpidem SL middle-of-nightZolpidem oral sprayZuranolone

Schedule V controlled substances (9)

PregabalinLacosamideBrivaracetamCenobamateEzogabineCannabidiolLasmiditanDiphenoxylateLacosamide ER

Second-generation antihistamines (8)

CetirizineLevocetirizineLoratadineDesloratadineFexofenadineAzelastineOlopatadineKetotifen

Second-generation antipsychotics (30)

ClozapineRisperidoneOlanzapineQuetiapineZiprasidoneAripiprazolePaliperidoneAsenapineIloperidoneLurasidoneBrexpiprazoleCariprazineLumateperoneMilsaperidonePimavanserinAmisulprideSulpirideAripiprazole lauroxil LAIAripiprazole lauroxil LAIAripiprazole monohydrate LAIAripiprazole monohydrate LAIAsenapine transdermalClozapine ODTClozapine oral suspensionPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIQuetiapine XRZiprasidone IM

Sedating medications (248)

MidazolamDexmedetomidineKetamineMethohexitalPentobarbitalRemimazolamTrazodoneQuetiapineMirtazapineZolpidemCyclobenzaprineTizanidineHydroxyzine HClOlanzapineAmitriptylineMeclizineTemazepamPromethazinePrimidoneDoxepinClozapineFentanylEszopiclonePhenobarbitalCarisoprodolSuvorexantChlorpromazineCyproheptadineRamelteonLumateperoneTriazolamEstazolamLemborexantDaridorexantThioridazineTasimelteonTrimipramineDoxylamineFlurazepamQuazepamGabapentinTramadolAlprazolamOxycodoneClonazepamLorazepamBuspironePregabalinBaclofenRisperidoneClonidineDiazepamMorphineMethocarbamolNortriptylineHydromorphoneProchlorperazinePaliperidoneMethadoneBuprenorphineBrexpiprazoleScopolamineImipramineZaleplonClobazamClorazepateClomipramineTapentadolDronabinolChlordiazepoxideCenobamateAsenapineLoxapineMetaxaloneChlorzoxazonePerampanelOrphenadrineHydrocodoneIloperidoneOxymorphoneOxazepamGabapentin enacarbilButorphanolCodeinePentazocineLevorphanolMeprobamateApomorphineMeperidineNalbuphineAcetaminophenZiconotideNabiloneBrompheniramineButalbitalChlorpheniramineDimenhydrinateDiphenhydramineGuanfacineSecobarbitalMetoprololSertralineCarvedilolDuloxetineEscitalopramCitalopramAtenololVenlafaxineOxybutyninLevetiracetamLamotriginePropranololParoxetineRopiniroleTopiramateDicyclomineLevocetirizineBenztropinePramipexoleCarbamazepineNebivololOxcarbazepineSotalolSolifenacinMetoclopramideLabetalolBisoprololHaloperidolDesvenlafaxineLurasidoneLacosamideTolterodineZiprasidoneVortioxetineAmantadineFluvoxamineZonisamideVilazodoneNadololFluphenazineTrihexyphenidylPerphenazineFesoterodineRasagilinePimavanserinDesloratadineEntacaponePhenytoinBrivaracetamEslicarbazepineMilnacipranRotigotineAcebutololEsketamineDesipramineSelegilineCannabidiolTrifluoperazineCetirizineHyoscyamineGepironeRufinamideFelbamatePindololThiothixeneCarteololIstradefyllineCarbidopaTiagabineOpicaponeMilsaperidoneEthosuximidePhenelzineTranylcyprominePimozideAprepitantLevodopaGranisetronProtriptylineZuranoloneNefazodoneAmoxapineMethsuximideVigabatrinFenfluramineRolapitantIsocarboxazidTrimethobenzamideStiripentolTolcaponeMolindoneFosphenytoinGanaxoloneDroperidolAmisulprideAlprazolam XRAmantadine ERAsenapine transdermalBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRClonidine ERClonidine ER suspensionClozapine ODTClozapine oral suspensionDexmedetomidine sublingualDoxepin low-dose (insomnia)Fluphenazine decanoate LAIFluvoxamine CRGuanfacine ERHaloperidol decanoate LAIHaloperidol injectionHydrocodone ER (q12h)Hydrocodone ER (q24h)Hydromorphone ERHydroxyzine IMLacosamide ERLamotrigine XRLorazepam injectionLoxapine inhaledMetoprolol succinate ERMorphine ER capsulesMorphine ER tabletsOxcarbazepine XROxybutynin EROxycodone CRPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIParoxetine CRPropranolol ERQuetiapine XRSelegiline transdermalTopiramate ERTopiramate ER (sprinkle)Tramadol ERVenlafaxine XRZiprasidone IMZolpidem CRZolpidem SLZolpidem SL middle-of-nightZolpidem oral spray

Seizure-threshold–lowering medications (54)

BupropionClozapineChlorpromazineOlanzapineQuetiapineTramadolMeperidineAmitriptylineClomipramineImipramineMaprotilineAmphetamineMethylphenidateTheophyllineCiprofloxacinLevofloxacinImipenemErtapenemMetronidazoleIsoniazidDiphenhydramineAminophyllineCocaineDalfampridineFlumazenilTiagabineAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)Bupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERClozapine ODTClozapine oral suspensionMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchMixed amphetamine salts (triple-bead)Mixed amphetamine salts XRQuetiapine XRTramadol ER

Selective estrogen receptor modulators (SERMs) (6)

RaloxifeneTamoxifenOspemifeneClomipheneBazedoxifeneToremifene

Selective serotonin reuptake inhibitors (SSRIs) (9)

SertralineEscitalopramFluoxetineCitalopramParoxetineFluvoxamineVilazodoneFluvoxamine CRParoxetine CR

Serotonin reuptake inhibitors (SRIs) (46)

TrazodoneSertralineTramadolDuloxetineEscitalopramFluoxetineCitalopramVenlafaxineAmitriptylineParoxetineNortriptylineDoxepinDesvenlafaxineVortioxetineFluvoxamineVilazodoneAtomoxetineChlorpromazineImipramineClomipramineLumateperoneMilnacipranDesipramineLevomilnacipranDextromethorphanProtriptylineNefazodoneAmoxapine8-OH-AmoxapineCentanafadineCocaineDesmethyl­ clomipramineDesmethyl­ sertralineHydroxy­ nefazodoneIbogaineNordoxepinNorfluoxetineNoribogaineTrimipramineZiprasidoneDoxepin low-dose (insomnia)Fluvoxamine CRParoxetine CRTramadol ERVenlafaxine XRZiprasidone IM

Serotonin-releasing agents (10)

FenfluramineMethylenedioxy­ methamphetamineAmphetamineMephedroneMethamphetamineAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)Mixed amphetamine salts (triple-bead)Mixed amphetamine salts XR

Serotonin–norepinephrine reuptake inhibitors (SNRIs) (6)

VenlafaxineDuloxetineDesvenlafaxineLevomilnacipranMilnacipranVenlafaxine XR

Sexual-dysfunction–associated medications (38)

SertralineFluoxetineParoxetineCitalopramEscitalopramFluvoxamineVenlafaxineDuloxetineClomipramineAmitriptylineRisperidonePaliperidoneHaloperidolFinasterideDutasterideSpironolactonePropranololMetoprololHydrochloro­ thiazideMorphineMethadoneLeuprolideBicalutamideDesvenlafaxineTamsulosinFluvoxamine CRHaloperidol decanoate LAIHaloperidol injectionMetoprolol succinate ERMorphine ER capsulesMorphine ER tabletsPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIParoxetine CRPropranolol ERVenlafaxine XR

Sleep medications (25)

ZolpidemEszopicloneZaleplonSuvorexantLemborexantDaridorexantRamelteonDoxepinTemazepamTriazolamEstazolamFlurazepamQuazepamDiphenhydramineDoxylamineTasimelteonGHB (Oxybate)SecobarbitalSeltorexantDoxepin low-dose (insomnia)Mixed-salt oxybatesZolpidem CRZolpidem SLZolpidem SL middle-of-nightZolpidem oral spray

Smoking-cessation medications (12)

BupropionVareniclineNicotine gumBupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERNicotine inhalerNicotine lozengeNicotine nasal sprayNicotine patch

Sodium-glucose cotransporter-2 (SGLT2) inhibitors (7)

EmpagliflozinDapagliflozinCanagliflozinErtugliflozinBexagliflozinSotagliflozinLuseogliflozin

Somatostatin analogs (3)

OctreotideLanreotidePaltusotine

Statins (7)

AtorvastatinRosuvastatinSimvastatinPravastatinLovastatinPitavastatinFluvastatin

Stevens–Johnson syndrome/toxic epidermal necrolysis (SJS/TEN)–associated drugs (32)

AllopurinolCarbamazepineOxcarbazepinePhenytoinPhenobarbitalLamotrigineDapsoneNevirapineZonisamideAbacavirArmodafinilFosphenytoinMeloxicamModafinilPiroxicamSulfamethoxazoleTrimethoprimValproic acidDiclofenacIbuprofenCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchDivalproex DRDivalproex ERDivalproex sprinkleLamotrigine XROxcarbazepine XRValproate sodium IV

Stimulants (41)

AmphetamineDextro­ amphetamineMethamphetamineLisdexamfetamineMethylphenidateDex­ methylphenidateCocaineModafinilArmodafinilSolriamfetolCaffeinePhentermineCathinoneMethylenedioxy­ pyrovaleroneMephedronePhendimetrazineAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)Dexmethylphenidate XRDextroamphetamine IR tabletsDextroamphetamine oral solutionDextroamphetamine patchDextroamphetamine spansuleMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchMixed amphetamine salts (triple-bead)Mixed amphetamine salts XRSerdexmethylphenidate

Substance-use treatment (25)

BupropionMethadoneVareniclineBuprenorphineNaltrexoneAcamprosateNicotine gumDisulfiramLofexidineNalmefeneBuprenorphine ER injectionBuprenorphine SC (weekly/monthly)Buprenorphine buccal filmBuprenorphine patchBuprenorphine/ naloxoneBupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERNaltrexone ER injectionNicotine inhalerNicotine lozengeNicotine nasal sprayNicotine patch

Sulfonamides (16)

SulfamethoxazoleAcetazolamideBumetanideCelecoxibChlorthalidoneDapsoneDarunavirFurosemideHydrochloro­ thiazideIndapamideMethazolamideProbenecidSulfasalazineSumatriptanSumatriptan SC injectionSumatriptan nasal

Sympatholytics (29)

MetoprololCarvedilolAtenololPropranololNebivololSotalolLabetalolBisoprololNadololAcebutololPindololCarteololPhenoxybenzaminePhentolamineGuanabenzMethyldopaClonidineDoxazosinGuanfacinePrazosinReserpineTerazosinClonidine ERClonidine ER suspensionGuanfacine ERMetoprolol succinate ERMoxonidinePropranolol ERRilmenidine

Sympathomimetics (57)

MethylphenidateMegestrolLisdexamfetamineOlopatadineModafinilAtomoxetineCyproheptadineArmodafinilDextro­ amphetamineDex­ methylphenidateAcebutololCetirizineCarteololSolriamfetolViloxazineOxymetazolineFilgrastimAmphetaminePhenylephrineMethamphetamineBisacodylCaffeineCathinoneCocaineDimenhydrinateMethylenedioxy­ pyrovaleroneMephedroneNeuropeptide YPseudoephedrineSennaDobutaminePhendimetrazineAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)DesglymidodrineDexmethylphenidate XRDextroamphetamine IR tabletsDextroamphetamine oral solutionDextroamphetamine patchDextroamphetamine spansuleMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchMixed amphetamine salts (triple-bead)Mixed amphetamine salts XR

Tardive dyskinesia treatments (3)

ValbenazineDeutetrabenazineTetrabenazine

Tetracyclic antidepressants (3)

MirtazapineMianserinMaprotiline

Tetracyclines (4)

DoxycyclineMinocyclineTetracyclineDemeclocycline

Thiazide diuretics (5)

Hydrochloro­ thiazideChlorthalidoneMetolazoneIndapamideChlorothiazide

Thiazolidinediones (3)

PioglitazoneRosiglitazoneLobeglitazone

Thrombolytics (3)

Tranexamic acidAlteplaseTenecteplase

Thrombosis-associated medications (57)

Ethinyl estradiolConjugated estrogensEstradiolTamoxifenRaloxifeneClomipheneTestosteroneLenalidomideTofacitinibUpadacitinibMegestrolMedroxy­ progesteroneNorethindroneTranexamic acidOspemifeneDrospirenoneLevonorgestrelProgesteroneAbrocitinibAndexanet alfaApixabanCelecoxibDabigatranDanazolDarbepoetin alfaDiclofenacDiflunisalEdoxabanEpoetin alfaEtodolacEverolimusFenoprofenFlurbiprofenIbuprofenIndomethacinKetoprofenKetorolacMeclofenamateMefenamic acidMeloxicamNabumetoneNaproxenOxaprozinPiroxicamRivaroxabanSalsalateSulindacTiclopidineTolmetinDiclofenac oral solutionDiclofenac topical gelDiclofenac topical patchEstradiol transdermalEstradiol vaginalLevonorgestrel IUDMedroxyprogesterone depotTestosterone cypionate

Thyroid hormones and analogs (3)

LevothyroxineLiothyronineThyroid, desiccated

Tocolytics (6)

TerbutalineAtosibanIndomethacinMagnesium sulfateNifedipineNifedipine ER (GITS)

Topical anti-inflammatory drugs (13)

ClobetasolMometasoneBetamethasoneFluocinonideFluorometholoneBromfenacHalobetasolCrisaboroleDiclofenacHydrocortisonePimecrolimusTacrolimusTriamcinolone

Topoisomerase inhibitors (4)

TopotecanDoxorubicinEtoposideIrinotecan

Trace amine-associated receptor 1 (TAAR1) agonists (1)

Ulotaront

Tricyclic antidepressants (TCAs) (10)

AmitriptylineImipramineClomipramineNortriptylineDesipramineDoxepinTrimipramineProtriptylineAmoxapineDoxepin low-dose (insomnia)

Triptans (9)

SumatriptanRizatriptanNaratriptanEletriptanZolmitriptanFrovatriptanAlmotriptanSumatriptan SC injectionSumatriptan nasal

Tuberculosis drugs (7)

RifampinEthambutolIsoniazidRifapentineCycloserineBedaquilinePyrazinamide

Tubular toxicity (acute tubular necrosis) (11)

GentamicinTobramycinAmikacinVancomycinAmphotericin BCisplatinTenofovirCidofovirNeomycinAdefovirFoscarnet

Tumor necrosis factor (TNF) inhibitors (3)

AdalimumabEtanerceptInfliximab

Tyrosine kinase inhibitors (TKIs) (25)

AcalabrutinibAlectinibBosutinibCeritinibCrizotinibDasatinibErlotinibIbrutinibImatinibLorlatinibNilotinibOsimertinibRegorafenibTucatinibVandetanibZanubrutinibAfatinibAsciminibCapmatinibDacomitinibFruquintinibGefitinibPonatinibQuizartinibRipretinib

Unavailable currently (31)

AceclidineAficamtenAjmalineAmisulprideAprindineAtosibanBetahistineBitopertinCibenzolineCisaprideClodronateCloxacillinDomperidoneEncainideEthacizineEthchlorvynolEtoricoxibEzogabineFlunitrazepamFlupentixolGlutethimideHeroinHydroquinidineIclepertinImrecoxibLorcaserinMelperonePhenibutReboxetineSermorelinTicarcillin

Uricosurics (2)

ProbenecidLesinurad

Urinary-retention–associated medications (38)

BenztropineTrihexyphenidylOxybutyninTolterodineSolifenacinDarifenacinTrospiumAmitriptylineImipramineClomipramineClozapineOlanzapineChlorpromazineDiphenhydramineChlorpheniraminePseudoephedrinePhenylephrineMorphineOxycodoneAtropineDicyclomineDoxepinFesoterodineGlycopyrrolateHydroxyzine HClHyoscyamineNortriptylineScopolamineAtropine eyedropsClozapine ODTClozapine oral suspensionDoxepin low-dose (insomnia)Glycopyrrolate inhaledHydroxyzine IMMorphine ER capsulesMorphine ER tabletsOxybutynin EROxycodone CR

Uterotonics (8)

CabergolineBromocriptineFezolinetantOxytocinDinoprostoneMethylergonovineMisoprostolCarboprost

Vascular endothelial growth factor (VEGF) inhibitors (4)

AfliberceptBevacizumabFaricimabRanibizumab

Vasodilators (34)

HydralazineNitroglycerinDoxazosinPrazosinMinoxidil oralPentoxifyllineGuanfacineMacitentanAmbrisentanRiociguatDipyridamoleBosentanPhenoxybenzaminePhentolamineAmyl nitriteAmlodipineClevidipineEpoprostenolFelodipineFenoldopamIsosorbide dinitrateIsosorbide mononitrateNicardipineNifedipineNitroprussideSelexipagSildenafilTadalafilTreprostinilVericiguatGuanfacine ERMinoxidil topicalNifedipine ER (GITS)Tadalafil (PAH)

Vasopressin agonists (5)

DesmopressinCannabidiolOxytocinTerlipressinVasopressin

Vasopressin antagonists (4)

TolvaptanAtosibanConivaptanDemeclocycline

Vasopressors (8)

MidodrineDroxidopaDobutamineNorepinephrineVasopressinDopamineEpinephrinePhenylephrine

Very long half-life drugs (80)

AmiodaroneHydroxy­ chloroquineDorzolamideDutasterideTerbinafineRaloxifeneDenosumabMedroxy­ progesteroneRisedronateBrinzolamideMefloquineZoledronic acidChloroquineMitotaneCholecalciferolErenumabFremanezumabGalcanezumabPyridoxineSiltuximabVandetanibAlirocumabTeriflunomideErgocalciferolLeflunomideCalcifediolAmphotericin BEvolocumabAdalimumabClodronateRomosozumabTocilizumabUmeclidiniumAlendronateNorfluoxetineInfliximabPentamidineRimonabantSarilumabDidesmethyl­ cariprazineLevothyroxineSemaglutideFingolimodRolapitantEndoxifenThyroid, desiccatedTamoxifenCyanocobalaminBicalutamideEnzalutamideMavacamtenAdenosylcobalaminMethylcobalaminRetatrutideEntecavirIsavuconazoniumIsavuconazoleFluoxetineDulaglutideTiotropiumTirzepatideClomipheneReserpinePerampanelEtanerceptUrsodiolTrametinibPyrimethamineThiamineDehydro­ aripiprazoleBrexpiprazoleIstradefyllineIcosapent ethylNetupitantPhenobarbitalBaloxavir marboxilAripiprazoleApalutamideProtriptylineDesmethyl­ sertraline

Very short half-life drugs (227)

ClevidipineSalvinorin ASuccinylcholineEpinephrineDobutamineDopamineMivacuriumNorepinephrineIsoproterenolNitroglycerinHeroinOxytocinFenoldopamEpoprostenolTetracaineProcaineEsmololRemifentanilTestosteroneFluorouracilEdrophoniumProtamine sulfateFosphenytoinAjmalineN,N-dimethyl­ tryptamineGlucagonPhentolamineAtosibanAtracuriumSodium thiosulfateAspirinVasopressinProgesteroneAldosteroneArticaineCisatracuriumPsilocybinMupirocinValacyclovirLinaclotideMidodrineMisoprostolPenicillin VNafcillinOxacillinNitrofurantoinDeferoxamineTropicamideCarbacholCloxacillinDimercaprolGHB (Oxybate)IV lipid emulsionMethicillinRetinolBenazeprilFolic acidDicloxacillinInsulin glulisineApomorphineMelatoninTravoprostTretinoinCapecitabineRemimazolamPramlintideTerlipressinPilocarpineOmeprazolePantoprazoleCephalexinInsulin lisproBumetanideLiothyronineGuaifenesinIsosorbide dinitrateLisdexamfetamineAzathioprineMolnupiravirLubiprostonePentoxifyllineRepaglinideRabeprazoleNiacinZaleplonCalcitonin (salmon)TeriparatideAcalabrutinibMeropenemDimethyl fumarateSelexipagPerindoprilDiroximel fumarateFlumazenilRemdesivirAndexanet alfaCocaineImipenemNeostigmineYohimbineChlorzoxazoneBelinostatRamelteonVecuroniumAmoxicillinEstradiolEsomeprazoleEnalaprilAmpicillinTasimelteonCefuroximeClavulanateRiboflavinMethsuximideOliceridineRocuroniumSacubitrilAllopurinolSpironolactoneInsulin aspartHydrocortisoneMethocarbamolLidocaineErythromycinLansoprazoleDexlansoprazoleNaloxoneGemfibrozilCefadroxilRivastigmineBethanecholNateglinideBalsalazideCromolynHeparinMercaptopurinePropylthiouracilIsoniazidAbacavirOpicaponeAlosetronLevodopaNizatidineChlorothiazideMolindoneMannitolPhysostigmineEdetate calcium disodiumPralidoximeRegular insulinAlfentanilPrilocaineCefdinirGlycopyrrolateAbaloparatideOctreotidePhytonadioneCefazolinFlunisolideLosartanFurosemideSimvastatinLatanoprostPravastatinDiclofenacIbuprofenOxybutyninNifedipineIpratropiumRamiprilBimatoprostOxcarbazepineTolterodineGentamicinCarisoprodolPyridostigmineTobramycinAcarboseClorazepateFamciclovirCimetidineCefepimeCaptoprilQuinaprilIvabradineSelegilineNicotine gumTranexamic acidMoexiprilCarbidopaCeftazidimeEthacrynic acidAmikacinTriamtereneAztreonamKetoprofenDeferipronePenicillamineIsocarboxazidTrofinetideVorinostatMefenamic acidSuccimerErgotamineDexmedetomidineNabiloneAceclidineAgmatineBiotinEncainideIndinavirJWH-018Methylenedioxy­ pyrovaleroneMephedroneMepivacaineMethyldopaMoclobemideMoricizineSugammadexCefotaximeCefoxitinGlycerinNystatinPenicillin GPiperacillinProcarbazineL-Theanine

Vesicular monoamine transporter 2 (VMAT2) inhibitors (6)

ValbenazineDeutetrabenazineTetrabenazineMethamphetamine[+]-α-HTBZReserpine

Vitamin D analogs (7)

ErgocalciferolCalcitriolCalcipotrieneCalcifediolParicalcitolCholecalciferolDoxercalciferol

Vitamin K antagonists (1)

Warfarin

Vitamins and minerals (32)

WarfarinErgocalciferolCalcitriolFolic acidRiboflavinCyanocobalaminNiacinCalcipotrieneCalcifediolParicalcitolDoxercalciferolThiamineAdenosylcobalaminα-TocopherolAscorbic acidBiotinCholecalciferolMenaquinoneMethylcobalaminPantothenic acidPhytonadionePyridoxineRetinol5-hydroxy­ tryptophanCholineFerrous sulfateL-MethylfolateMagnesium oxideNicotinamidePyridoxal-5'- phosphateTryptophanCreatine

Wake-promoting drugs (32)

ModafinilArmodafinilSolriamfetolPitolisantAmphetamineDextro­ amphetamineMethylphenidateMethamphetamineCaffeineAmphetamine XR suspensionAmphetamine XR-ODTAmphetamine racemic (1:1)Dextroamphetamine IR tabletsDextroamphetamine oral solutionDextroamphetamine patchDextroamphetamine spansuleMethylphenidate CDMethylphenidate ER (OROS)Methylphenidate ER (Relexxii)Methylphenidate ER chewableMethylphenidate ER evening-dosedMethylphenidate ER suspensionMethylphenidate LAMethylphenidate SRMethylphenidate XR (Adhansia)Methylphenidate XR (Aptensio)Methylphenidate XR-ODTMethylphenidate chewableMethylphenidate oral solutionMethylphenidate patchMixed amphetamine salts (triple-bead)Mixed amphetamine salts XR

Weight-gain–associated medications (162)

OlanzapineClozapineMegestrolPrednisoneQuetiapineInsulin glargineMirtazapineTriamcinoloneMethyl­ prednisolonePioglitazoneInsulin lisproInsulin aspartHydrocortisoneInsulin detemirInsulin degludecDexamethasoneBudesonideFludrocortisoneChlorpromazineCyproheptadineThioridazineBexagliflozinInsulin glulisinePramlintideSotagliflozinGlipizidePregabalinGlimepirideRisperidoneAmitriptylineParoxetineDoxepinPaliperidoneBrexpiprazoleMedroxy­ progesteroneGlyburideImipramineClomipramineLumateperoneAsenapineIloperidonePhenelzineVigabatrinTrimipramineIsocarboxazidLithiumAtenololGabapentinMetoprololPrednisolonePropranololRosiglitazoneValproic acidTrazodoneSertralineCarvedilolEscitalopramClonazepamFluoxetineCitalopramHydroxyzine HClAripiprazoleLevocetirizinePromethazineCarbamazepineNebivololPrimidoneNortriptylineSotalolLabetalolBisoprololHaloperidolLurasidoneProchlorperazineCariprazineVortioxetinePhenobarbitalFluvoxamineRepaglinideVilazodoneNadololFluphenazinePerphenazineClobazamNateglinidePimavanserinDesloratadinePhenytoinBrivaracetamDronabinolEslicarbazepineMilnacipranCenobamateAcebutololLoxapinePerampanelEsketamineDesipramineCannabidiolTrifluoperazineCetirizineGabapentin enacarbilGepironeRufinamidePindololThiothixeneCarteololTiagabineMilsaperidoneEthosuximideTranylcyprominePimozideProtriptylineZuranoloneNefazodoneAmoxapineMethsuximideFenfluramineDoxylamineTrimethobenzamideMolindoneFosphenytoinGanaxoloneDroperidolAmisulprideNabilonePentobarbitalAripiprazole lauroxil LAIAripiprazole lauroxil LAIAripiprazole monohydrate LAIAripiprazole monohydrate LAIAsenapine transdermalCarbamazepine ER (Equetro)Carbamazepine ER capsulesCarbamazepine XRClozapine ODTClozapine oral suspensionDivalproex DRDivalproex ERDivalproex sprinkleDoxepin low-dose (insomnia)Fluphenazine decanoate LAIFluvoxamine CRGlipizide ERHaloperidol decanoate LAIHaloperidol injectionHydrocortisone topicalHydroxyzine IMInsulin glargine U-300Lithium ERLoxapine inhaledMedroxyprogesterone depotMetoprolol succinate ERPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIPaliperidone palmitate LAIParoxetine CRPropranolol ERQuetiapine XRTriamcinolone injectionValproate sodium IV

Weight-loss medications (26)

PhentermineBupropionLiraglutideLorcaserinNaltrexoneOrforglipronPhendimetrazineRetatrutideRimonabantSemaglutideSetmelanotideTirzepatideTopiramateBupropion SRBupropion SR (smoking cessation)Bupropion XLBupropion XL 450 mgBupropion hydrobromide ERLiraglutide (obesity)Naltrexone ER injectionSemaglutide (obesity)Semaglutide oralSemaglutide oral (obesity)Tirzepatide (obesity)Topiramate ERTopiramate ER (sprinkle)

Xanthine oxidase inhibitors (2)

AllopurinolFebuxostat