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Not available in the U.S.

Hydroquinidine

SERECOR

What it isDihydro derivative of quinidine, a class IA sodium channel blocker; Brugada syndrome and arrhythmia.

Why this oneAlong with quinidine it is one of the few drugs that suppresses ventricular fibrillation in Brugada syndrome.

What limits itQT prolongation and cinchonism as for quinidine. Not US-approved.

FDA-approved for

Off-label

NO BOXED WARNINGS

Principal riskQT prolongation and cinchonism

Classes and tags

Clinical profile

Direct muscarinic antagonism0 / 4

Mechanism of action: Hydroquinidine ballicule

Hydroquinidine ballicule: receptor binding, kinetics and half-life diagram

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