Ballicules.com

Relebactam

in RECARBRIO

What it isA diazabicyclooctane beta-lactamase inhibitor paired with imipenem-cilastatin.

Why this oneIt shields imipenem from KPC carbapenemases and derepressed AmpC, recovering activity against resistant Pseudomonas and Enterobacterales.

What limits itMetallo-beta-lactamases and many class D enzymes remain outside its reach.

NO BOXED WARNINGS

Classes and tags

Clinical profile

Direct muscarinic antagonism0 / 4

Mechanism of action: Relebactam ballicule

Relebactam ballicule: receptor binding, kinetics and half-life diagram

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