Not available in the U.S.
Celiprolol
What it isCardioselective beta-1 adrenergic antagonist with partial beta-2 agonist and mild vasodilatory activity.
Why this oneUsed outside the US for hypertension and shown to reduce arterial events in vascular Ehlers-Danlos syndrome.
What limits itP-glycoprotein and OATP substrate whose absorption is reduced by food and by transporter-modulating drugs.
NO BOXED WARNINGS
Principal riskNo FDA boxed warning.
Classes and tags
Clinical profile
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Self-check
- In which inherited vascular condition has celiprolol reduced arterial events?
Vascular Ehlers-Danlos syndrome. - How does food affect celiprolol absorption?
Reduces it.