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Lobeglitazone

DUVIE

What it isThiazolidinedione PPAR-gamma agonist that improves peripheral insulin sensitivity.

Why this oneApproved in South Korea (Duvie) for type 2 diabetes, delivering glitazone-class glycemic benefit at low milligram doses.

What limits itShares TZD-class risks of fluid retention, heart failure exacerbation, weight gain and fracture, and is not FDA-approved.

NO BOXED WARNINGS

Principal riskNo FDA boxed warning.

Classes and tags

Clinical profile

Direct muscarinic antagonism0 / 4

Mechanism of action: Lobeglitazone ballicule

Lobeglitazone ballicule: receptor binding, kinetics and half-life diagram

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