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Tocainide

TONOCARD

What it isOral class IB antiarrhythmic, a lidocaine analogue; withdrawn.

Why this oneIt offered oral lidocaine-like activity for ventricular arrhythmia.

What limits itAgranulocytosis and pulmonary fibrosis ended its use.

FDA-approved for

⚠ BOXED WARNINGS

Classes and tags

Clinical profile

Direct muscarinic antagonism0 / 4

Mechanism of action: Tocainide ballicule

Tocainide ballicule: receptor binding, kinetics and half-life diagram

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