Ballicules.com
Not available in the U.S.

Ajmaline

GILURYTMAL

Ajmaline ballicule: receptor binding, kinetics and half-life diagram
Mechanism of action: Ajmaline ballicule

What it isClass IA sodium channel blocker; arrhythmias and Brugada provocation testing.

Why this oneMain modern use: unmasks the Brugada ECG pattern within minutes.

What limits itTesting itself risks proarrhythmia; resuscitation must be available. Not US-approved.

Ajmaline molecular structure (skeletal formula)
Molecular structure: Ajmaline

Used for

NO BOXED WARNINGS

Principal riskProarrhythmia during the test itself, so it is done with resuscitation available

Classes and tags

Clinical profile

Therapeutic safety burden3 / 4
Sedation liability0 / 4
QT / Torsades4 / 4
Direct muscarinic antagonism0 / 4
Embryofetal risk2 / 4

Defining liabilityProarrhythmia, QT prolongation and AV block requiring continuous ECG

Open Ajmaline in the interactive console ↗

Self-check