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Mechanisms
› GABA-A PAM
GABA-A PAM
GABA-A receptor positive allosteric modulator
Inhibition of neuron firing
➔ antiepileptic effects
➔ sedation
➔ ataxia
➔ anterograde amnesia
➔ muscle relaxation
Drugs with this mechanism (61)
Allopregnanolone
α-hydroxy alprazolam
Alprazolam
Zolpidem CR
Amobarbital
Androstanediol
Brexanolone
Butabarbital
Butalbital
Carisoprodol
Cenobamate
Chlordiazepoxide
Clobazam
Clonazepam
Desflurane
Diazepam
Zolpidem SL
Estazolam
Eszopiclone
Ethanol
Ethchlorvynol
Etomidate
Felbamate
Flunitrazepam
Flurazepam
Ganaxolone
Glutethimide
Halazepam
Zolpidem SL middle-of-night
Isoflurane
Lorazepam
Lorazepam injection
Meprobamate
Methaqualone
Methohexital
Midazolam
Norclobazam
Nordiazepam
Oxazepam
Pentobarbital
Phenobarbital
Pregnanolone
Primidone
Propofol
Quazepam
Topiramate ER (sprinkle)
Remimazolam
Secobarbital
Sevoflurane
Stiripentol
Temazepam
THDOC
Thiopental
Topiramate
Topiramate ER
Triazolam
Alprazolam XR
Zaleplon
Zolpidem
Zolpidem oral spray
Zuranolone
All mechanisms
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