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Nalmefene auto-injector

ZURNAI

Nalmefene auto-injector ballicule: receptor binding, kinetics and half-life diagram
Mechanism of action: Nalmefene auto-injector ballicule

NO BOXED WARNINGS

Clinical profile

Therapeutic safety burden1 / 4
Overdose danger1 / 4
Weight-gain liability0 / 4
Sedation liability0 / 4
QT / Torsades0 / 4
Direct muscarinic antagonism0 / 4
Embryofetal risk2 / 4

Legacy pregnancy categoryC

Defining liabilityUsually well tolerated; abrupt opioid withdrawal can be severe and prolonged.

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