Androgen receptor antagonist
- Blocks androgen-driven prostate cancer growth
- Gynecomastia, hot flashes, fatigue
- Newer agents lower seizure threshold
Drugs with this mechanism (4)
- Apalutamide — Androgen-receptor antagonist for prostate cancer; GABA-A effects give seizure risk.
- Bicalutamide — Androgen-receptor antagonist for prostate cancer.
- Darolutamide — Androgen-receptor inhibitor for advanced prostate cancer; minimal CNS penetration.
- Enzalutamide — Androgen-receptor antagonist for prostate cancer; GABA-A effects give seizure risk.
All mechanisms · Open the interactive console ↗