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5-HT2A inverse agonist
5-HT2A serotonin receptor inverse agonist
Pimavanserin for Parkinson disease psychosis
Drugs with this mechanism (2)
Norclozapine
— Active clozapine metabolite; M1 agonist implicated in some clozapine effects.
Pimavanserin
— Selective 5-HT2A inverse agonist; the first drug for Parkinson psychosis, no D2 blockade.
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